SCHEMBL11098527

SCHEMBL11098527

CC(C(=O)O)C(Br)C(=O)c1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
CYP1A2 P05177 1/20 0.47
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
POLB P06746 2/20 0.43
CES2 O00748 3/20 0.42
CES1 P23141 3/20 0.42
SRD5A2 P31213 1/20 0.41
TRPA1 O75762 2/20 0.41
GSK3B P49841 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
MEN1 O00255 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11204713 0.83 ALDH1A1 (0.47) ALDH1A1CYP1A2TSHRCES2CES1
SCHEMBL6417147 0.83 TRPA1 (0.47) ALDH1A1CYP1A2ALOX15TSHRCES2
SCHEMBL634548 0.79 CES2 (0.50) ALDH1A1CYP1A2ALOX15TSHRCES2
SCHEMBL28117241 0.78 ALOX15 (0.48) ALDH1A1ALOX15TSHRPOLBCES2
SCHEMBL8683450 0.77 ALOX15 (0.52) ALDH1A1ALOX15TSHRPOLBCES2
SCHEMBL28750316 0.75 ALDH1A1 (0.47) ALDH1A1CYP1A2TSHRTRPA1KMT2A
SCHEMBL10832344 0.75 HDAC3 (0.49) ALDH1A1ALOX15TSHRPOLBCES2
SCHEMBL2625462 0.74 CES2 (0.54) ALDH1A1ALOX15TSHRCES2CES1
SCHEMBL20995299 0.74 CES2 (0.54) ALDH1A1ALOX15TSHRCES2CES1
SCHEMBL3424507 0.74 GSK3B (0.61) ALDH1A1ALOX15TSHRCES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0037710-B1 THIAZOLE DERIVATIVES JOHN WYETH & BROTHER LIMITED (GB) 1984-08-01 EP disclosed
US-4385059-A 4-(4-CHLOROPHENYL)-2-(4-HYDROXYPHENYL)THIAZOLE-5-ACETIC ACID JOHN WYETH AND BROTHER LIMITED (GB) 1983-05-24 US disclosed
EP-0037710-A1 Thiazole derivatives JOHN WYETH & BROTHER LIMITED (GB) 1981-10-14 EP disclosed