SCHEMBL11098569

SCHEMBL11098569

COc1ccc(C(O)CNCc2ccccc2Br)cc1OC

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.54
ADRB2 P07550 5/20 0.50
DRD2 P14416 3/20 0.47
DRD3 P35462 3/20 0.47
ADRB1 P08588 3/20 0.47
DRD1 P21728 2/20 0.47
DRD4 P21917 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
SLC6A4 P31645 2/20 0.46
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
SLC22A1 O15245 1/20 0.46
CHRM2 P08172 1/20 0.46
CYP3A4 P08684 1/20 0.46
CHRM1 P11229 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
OPRM1 P35372 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11102216 0.88 MEN1 (0.59) OPRK1ADRB2DRD2DRD3ADRB1
SCHEMBL8907016 0.86 ADRB2 (0.51) OPRK1ADRB2DRD2DRD3ADRB1
SCHEMBL11099823 0.85 ADRB2 (0.50) OPRK1ADRB2DRD2DRD3ADRB1
SCHEMBL8905807 0.82 OPRK1 (0.48) OPRK1ADRB2DRD2DRD3ADRB1
SCHEMBL8993333 0.82 ALDH1A1 (0.48) OPRK1ADRB2DRD2DRD3ADRB1
SCHEMBL11099951 0.82 ADRB2 (0.61) OPRK1ADRB2DRD2DRD3ADRB1
SCHEMBL11268795 0.80 ALDH1A1 (0.60) ADRB2DRD2DRD3ADRB1DRD1
SCHEMBL8906035 0.78 OPRK1 (0.44) OPRK1ADRB2DRD2DRD3ADRB1
SCHEMBL178900 0.78 MEN1 (0.59) OPRK1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL8906047 0.75 ADRB3 (0.60) OPRK1ADRB2ADRB1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0040956-B1 8-SUBSTITUTED 4-(3,4-DIHYDROXYPHENYL)-1,2,3,4-TETRAHYDROISOQUINOLINES SMITHKLINE BECKMAN CORPORATION (US) 1984-10-31 EP disclosed
US-4340600-A Renal dilating methods and compositions using 4-(3,4-dihydroxyphenyl)-1,2,3,4-tetrahydroisoquinolines SMITHKLINE CORPORATION (US) 1982-07-20 US disclosed
EP-0040956-A1 8-Substituted 4-(3,4-dihydroxyphenyl)-1,2,3,4-tetrahydroisoquinolines SMITHKLINE BECKMAN CORPORATION (US) 1981-12-02 EP disclosed