SCHEMBL11102011

SCHEMBL11102011

CC(C)(C)c1ccc(SCCBr)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
HRH3 Q9Y5N1 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
HRH4 Q9H3N8 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.46
TSHR P16473 1/20 0.39
LMNA P02545 2/20 0.38
TYR P14679 1/20 0.38
MITF O75030 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SLC2A1 P11166 1/20 0.35
MAPK1 P28482 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10599472 0.87 ALDH1A1 (0.57) ALDH1A1NPC1RAB9AL3MBTL1HRH3
SCHEMBL2329783 0.86 ALDH1A1 (0.46) ALDH1A1NPC1RAB9AL3MBTL1HRH3
SCHEMBL5168465 0.83 ALDH1A1 (0.53) ALDH1A1NPC1RAB9AL3MBTL1HRH3
SCHEMBL11196940 0.79 ALDH1A1 (0.50) ALDH1A1NPC1RAB9AL3MBTL1HRH3
SCHEMBL10684156 0.79 ALDH1A1 (0.55) ALDH1A1NPC1RAB9AL3MBTL1HRH3
SCHEMBL2161163 0.79 ALDH1A1 (0.55) ALDH1A1NPC1RAB9AL3MBTL1HRH3
SCHEMBL7058481 0.78 MAOA (0.50) ALDH1A1NPC1RAB9AL3MBTL1HRH3
SCHEMBL10471246 0.76 ALDH1A1 (0.51) ALDH1A1NPC1RAB9AL3MBTL1HRH3
SCHEMBL16301153 0.76 NPC1 (0.47) ALDH1A1NPC1RAB9AL3MBTL1HRH3
SCHEMBL25934909 0.76 ALDH1A1 (0.47) ALDH1A1NPC1RAB9AL3MBTL1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0034784-B1 3,4,5-TRIHYDROXYPIPERIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICINES AND IN ANIMAL FEEDING BAYER AG (DE) 1984-07-25 EP disclosed
US-4407809-A N-phenoxy(or thio)hydrocarbon 3,4,5-trihydroxypiperidine derivatives, their use in medicine and in animal nutrition BAYER AKTIENGESELLSCHAFT (DE) 1983-10-04 US disclosed