SCHEMBL11113044

SCHEMBL11113044

CCCCCCc1ccc(OC(=O)NCCN2CCCC2)nc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.44
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
BCHE P06276 2/20 0.43
ACHE P22303 2/20 0.43
THRA P10827 2/20 0.42
THRB P10828 2/20 0.42
KDM4E B2RXH2 1/20 0.42
SPHK1 Q9NYA1 1/20 0.42
CYP2D6 P10635 1/20 0.41
GLA P06280 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11118776 0.90 HRH3 (0.47) HRH3BCHEACHECYP2D6
SCHEMBL11131225 0.80 KCNH2 (0.41) THRATHRBKDM4ECYP2D6L3MBTL1
SCHEMBL11118198 0.76 HRH3 (0.46) HRH3ACHECYP2D6
SCHEMBL11116202 0.76 ALDH1A1 (0.45) THRATHRBKDM4ECYP2D6L3MBTL1
SCHEMBL11114098 0.74 HRH3 (0.50) HRH3ACHECYP2D6
SCHEMBL11113046 0.74 HRH3 (0.50) HRH3ACHECYP2D6
SCHEMBL11110142 0.74 GAA (0.46) BCHEKDM4EL3MBTL1
SCHEMBL11911916 0.72 HRH3 (0.46) HRH3CYP2D6
Hydrochloric Acid SCHEMBL4251038 0.71 HRH3 (0.47) HRH3CYP2D6
SCHEMBL9367313 0.71 MGLL (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0123700-A1 Substituted picolinic acids, processes for their preparation, their use, and pharmaceutical preparations containing them Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1984-11-07 EP disclosed