SCHEMBL11116202

SCHEMBL11116202

CCCCc1ccc(OC(=O)NCCN(C)C)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
CYP1A2 P05177 2/20 0.45
MAPT P10636 2/20 0.45
NFKB1 P19838 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
CYP3A4 P08684 1/20 0.45
PKM P14618 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
THPO P40225 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
KMT2A Q03164 1/20 0.45
HIF1A Q16665 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
THRA P10827 2/20 0.41
THRB P10828 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11110142 0.86 GAA (0.46) ALDH1A1CYP1A2MAPTNFKB1KDM4E
SCHEMBL11131225 0.85 KCNH2 (0.41) ALDH1A1CYP1A2MAPTNFKB1KDM4E
SCHEMBL11120268 0.81 ALDH1A1 (0.40) ALDH1A1CYP1A2KDM4ETHRATHRB
SCHEMBL11110055 0.79 ALDH1A1 (0.45) ALDH1A1CYP1A2MAPTNFKB1KDM4E
SCHEMBL11118776 0.78 HRH3 (0.47) MAPTCYP2D6
SCHEMBL11114735 0.77 ALDH1A1 (0.54) ALDH1A1CYP1A2MAPTNFKB1KDM4E
SCHEMBL11114279 0.76 ALDH1A1 (0.60) ALDH1A1CYP1A2MAPTNFKB1KDM4E
SCHEMBL11113044 0.76 HRH3 (0.44) KDM4EL3MBTL1THRATHRBCYP2D6
SCHEMBL11116141 0.76 ACACB (0.41) SIGMAR1ATMACACB
SCHEMBL11115121 0.75 NFKB1 (0.55) ALDH1A1CYP1A2MAPTNFKB1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0123700-A1 Substituted picolinic acids, processes for their preparation, their use, and pharmaceutical preparations containing them Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1984-11-07 EP disclosed