SCHEMBL11114977

SCHEMBL11114977

O=C(O)C1Oc2ccc(N3CCCC3=O)cc2O1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
HPGD P15428 6/20 0.51
CYP2C19 P33261 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
NPC1 O15118 6/20 0.43
RAB9A P51151 5/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
KMT2A Q03164 4/20 0.43
TSHR P16473 3/20 0.43
MEN1 O00255 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GAA P10253 1/20 0.43
GRK2 P25098 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
TP53 P04637 1/20 0.42
MAPK1 P28482 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11114610 0.82 ALDH1A1 (0.47) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4
SCHEMBL11110414 0.82 ALDH1A1 (0.45) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4
SCHEMBL11117922 0.74 LMNA (0.63) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4
SCHEMBL10876568 0.74 CMA1 (0.56) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4
SCHEMBL11118270 0.70 CYP17A1 (0.46) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4
SCHEMBL11118161 0.70 ALDH1A1 (0.45) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4
SCHEMBL11142367 0.70 ALDH1A1 (0.74) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4
SCHEMBL11110045 0.70 CMA1 (0.54) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4
SCHEMBL70639 0.70 ALDH1A1 (1.00) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4
SCHEMBL12445273 0.69 LMNA (0.51) ALDH1A1HPGDCYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0106988-A1 Pharmacologically active lactam derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1984-05-02 EP claimed
EP-0106988-A1 Pharmacologically active lactam derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1984-05-02 EP disclosed