SCHEMBL11116639

SCHEMBL11116639

O=CC(=O)OCCc1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.69
AKR1B10 O60218 5/20 0.65
AKR1B1 P15121 5/20 0.65
MAOB P27338 1/20 0.58
ALOX5 P09917 4/20 0.54
CYP3A4 P08684 3/20 0.54
MAPK1 P28482 3/20 0.54
HSD17B10 Q99714 3/20 0.54
TDP1 Q9NUW8 3/20 0.54
ALOX15 P16050 2/20 0.54
ALOX12 P18054 2/20 0.54
ESR1 P03372 2/20 0.54
ALDH1A1 P00352 2/20 0.54
HPGD P15428 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
TP53 P04637 2/20 0.54
TSHR P16473 2/20 0.54
HIF1A Q16665 2/20 0.54
TTR P02766 2/20 0.54
LMNA P02545 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3482701 0.86 HCAR2 (0.89) HCAR2AKR1B10AKR1B1MAOBALOX5
SCHEMBL573377 0.86 HCAR2 (0.89) HCAR2AKR1B10AKR1B1MAOBALOX5
SCHEMBL9860306 0.86 HCAR2 (0.89) HCAR2AKR1B10AKR1B1MAOBALOX5
SCHEMBL40718 0.83 THRB (0.67) HCAR2AKR1B10AKR1B1MAOBALOX5
SCHEMBL4672346 0.83 HCAR2 (0.67) HCAR2AKR1B10AKR1B1MAOBALOX5
SCHEMBL23542545 0.83 HCAR2 (0.67) HCAR2AKR1B10AKR1B1MAOBALOX5
Phenylethyl Fumarate SCHEMBL573379 0.81 HCAR2 (1.00) HCAR2AKR1B10AKR1B1MAOBALOX5
Phenylethyl Fumarate SCHEMBL27750209 0.81 HCAR2 (1.00) HCAR2AKR1B10AKR1B1MAOBALOX5
SCHEMBL23343675 0.81 HCAR2 (0.75) HCAR2AKR1B10AKR1B1MAOBALOX5
Phenylethyl Fumarate SCHEMBL573376 0.81 HCAR2 (1.00) HCAR2AKR1B10AKR1B1MAOBALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2852374-B1 PROCESS FOR DYEING KERATIN FIBRES COMPRISING A DYE/PIGMENT, A PHOTOACTIVE COMPOUND AND A LIGHT SOURCE OREAL (FR) 2019-08-21 EP claimed
EP-2852374-A1 PROCESS FOR DYEING KERATIN FIBRES COMPRISING A DYE/PIGMENT, A PHOTOACTIVE COMPOUND AND A LIGHT SOURCE L'Oréal (FR) 2015-04-01 EP claimed
WO-2013174871-A1 PROCESS FOR DYEING KERATIN FIBRES COMPRISING A DYE/PIGMENT, A PHOTOACTIVE COMPOUND AND A LIGHT SOURCE L'OREAL (FR) 2013-11-28 WO claimed
WO-2020067457-A1 CONDENSED-CYCLIC COMPOUND 武田薬品工業株式会社 2020-04-02 WO disclosed
WO-2020067455-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 2020-04-02 WO disclosed
WO-2020067456-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 2020-04-02 WO disclosed
WO-2020059892-A1 INSULIN-PRODUCING CELLS 武田薬品工業株式会社 2020-03-26 WO disclosed
WO-2019189555-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 2019-10-03 WO disclosed
WO-2019189553-A1 HETEROCYCLIC COMPOUND 国立大学法人京都大学 2019-10-03 WO disclosed
WO-2019151269-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 2019-08-08 WO disclosed
EP-0106652-A1 Beta-lactam compounds and production thereof SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1984-04-25 EP disclosed