SCHEMBL1111708

SCHEMBL1111708

c1ccc(C(C2CCCCC2)N2CC[N]CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.57
OPRD1 P41143 4/20 0.57
OPRK1 P41145 4/20 0.57
OPRL1 P41146 3/20 0.57
CYP17A1 P05093 1/20 0.45
IDO1 P14902 2/20 0.42
CACNA2D1 P54289 3/20 0.41
CACNA1B Q00975 3/20 0.41
CACNB1 Q02641 3/20 0.41
CACNA1C Q13936 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
KCNA5 P22460 2/20 0.41
CYP2C19 P33261 2/20 0.41
KCNH2 Q12809 2/20 0.41
KCNE1 P15382 1/20 0.41
CHRM3 P20309 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7054929 0.86 OPRM1 (0.63) OPRM1OPRD1OPRK1OPRL1CYP17A1
SCHEMBL8124509 0.81 OPRD1 (0.57) OPRM1OPRD1OPRK1OPRL1CYP17A1
SCHEMBL12508362 0.81 OPRM1 (0.57) OPRM1OPRD1OPRK1OPRL1CYP17A1
SCHEMBL645116 0.78 OPRM1 (0.45) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL28554103 0.77 OPRM1 (0.57) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL20804476 0.76 ATM (0.52) OPRM1OPRD1OPRK1OPRL1
SCHEMBL492900 0.74 OPRM1 (0.50) OPRM1OPRD1OPRK1OPRL1IDO1
SCHEMBL20804659 0.74 CHRM3 (0.60) OPRM1OPRD1OPRK1OPRL1CYP1A2
SCHEMBL20804660 0.74 MAOB (0.61) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL644900 0.73 OPRM1 (0.49) OPRM1OPRD1OPRK1OPRL1CACNA2D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2279174-A2 ARYLSULFONAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF USE Genentech, Inc. (US) 2011-02-02 EP disclosed
WO-2009143246-A2 ARYLSULFONAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF USE GENENTECH, INC. (US) 2009-11-26 WO disclosed