SCHEMBL28554103

SCHEMBL28554103

O=C(O)N1CCN(C(c2ccccc2)C2CCCCC2)CC1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.57
OPRD1 P41143 2/20 0.57
OPRK1 P41145 2/20 0.57
OPRL1 P41146 2/20 0.57
CACNA2D1 P54289 5/20 0.56
CACNA1B Q00975 5/20 0.56
CACNB1 Q02641 5/20 0.56
CACNA1C Q13936 4/20 0.56
CNR1 P21554 3/20 0.55
CNR2 P34972 3/20 0.55
NPSR1 Q6W5P4 2/20 0.54
HTT P42858 1/20 0.54
CHRM3 P20309 4/20 0.53
TSHR P16473 1/20 0.50
KDM4E B2RXH2 1/20 0.49
MAPT P10636 1/20 0.49
HPGD P15428 1/20 0.49
KMT2A Q03164 1/20 0.49
ALDH1A1 P00352 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20804660 0.87 MAOB (0.61) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL7054929 0.82 OPRM1 (0.63) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL23293370 0.82 CACNA2D1 (0.51) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL643105 0.80 ALDH1A1 (0.55) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL20804479 0.79 SLC6A4 (0.52) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL12508362 0.77 OPRM1 (0.57) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL1111708 0.77 OPRM1 (0.57) OPRM1OPRD1OPRK1OPRL1CACNA2D1
SCHEMBL8124509 0.77 OPRD1 (0.57) OPRM1OPRD1OPRK1OPRL1CACNA2D1
Trifluoroacetic Acid SCHEMBL26980890 0.76 OPRD1 (0.56) OPRM1OPRD1OPRK1OPRL1CACNA2D1
Trifluoroacetic Acid SCHEMBL23293527 0.76 OPRD1 (0.56) OPRM1OPRD1OPRK1OPRL1CACNA2D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112585139-B Naphthyridinone compounds as T cell activators 百时美施贵宝公司 2023-12-01 CN disclosed
CN-112585139-A Nalidinone compounds as T cell activators 百时美施贵宝公司 2021-03-30 CN disclosed