SCHEMBL11112840

SCHEMBL11112840

CC(=O)n1cc2c3c(ccc(Cl)c31)C(=O)CC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.35
HSD17B10 Q99714 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
TYMS P04818 1/20 0.33
HSD17B1 P14061 2/20 0.32
PBRM1 Q86U86 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
BAZ2B Q9UIF8 1/20 0.31
USP2 O75604 1/20 0.31
S100A4 P26447 1/20 0.31
CYP1A2 P05177 1/20 0.31
POLB P06746 1/20 0.31
ERCC1 P07992 1/20 0.31
MAPT P10636 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11110418 0.78 NOTUM (0.31) NOTUMHSD17B10MEN1KMT2AKDM4E
SCHEMBL11117091 0.71 ALDH1A1 (0.33) ALDH1A1
SCHEMBL19216725 0.64 TYMS (0.40) MEN1KMT2AALDH1A1TYMSUSP2
SCHEMBL30067557 0.63 TYMS (0.57) HSD17B10MEN1KMT2AKDM4EALDH1A1
Acetic Acid SCHEMBL28550221 0.63 SRD5A1 (0.58) NOTUMHSD17B10HSD17B1CASP1CASP7
SCHEMBL11109712 0.62 CASP1 (0.36) HSD17B10MEN1KMT2ATYMSHSD17B1
SCHEMBL21948632 0.60 TYMS (0.53) HSD17B10MEN1KMT2AKDM4EALDH1A1
SCHEMBL6625286 0.60 CNR1 (0.34) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL8253223 0.59 NPC1 (0.61) HSD17B10HSD17B1PBRM1CASP1CASP7
SCHEMBL8283186 0.57 CASP1 (0.50) HSD17B10HSD17B1PBRM1CASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033767-B1 INDOLOBENZOXAZINES, PROCESSES FOR PREPARING AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME MERCK & CO. INC. (US) 1984-06-27 EP disclosed
EP-0033767-A1 Indolobenzoxazines, processes for preparing and pharmaceutical compositions containing the same MERCK & CO. INC. (US) 1981-08-19 EP disclosed
US-4238486-A TREATING HYPERTENSION AND PARKINSON*S DISEASE MERCK & CO., INC. (US) 1980-12-09 US disclosed