SCHEMBL11119002

SCHEMBL11119002

COc1ccc(C2(C(=O)O)CCNCC2C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.42
TET3 O43151 1/20 0.40
KMT2A Q03164 1/20 0.40
FBXL19 Q6PCT2 1/20 0.40
CXXC5 Q7LFL8 1/20 0.40
TET1 Q8NFU7 1/20 0.40
KDM2B Q8NHM5 1/20 0.40
CXXC4 Q9H2H0 1/20 0.40
KDM2A Q9Y2K7 1/20 0.40
ATM Q13315 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
THRB P10828 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
MMP3 P08254 1/20 0.38
MMP10 P09238 1/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11118224 0.84 OPRM1 (0.42) HSD11B1
SCHEMBL21119266 0.84 OPRM1 (0.42) HSD11B1
SCHEMBL8175346 0.78 CHRNA1 (0.43) ATML3MBTL1CHRNB2CHRNB4CHRNA3
SCHEMBL14232738 0.75 OPRM1 (0.40) HSD11B1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL16058193 0.75 KMT2A (0.57) TET3KMT2AFBXL19CXXC5TET1
SCHEMBL11094114 0.72 OPRM1 (0.60)
SCHEMBL11079554 0.72 HSD11B1 (0.47) HSD11B1TET3KMT2AFBXL19CXXC5
SCHEMBL378469 0.72 HSD11B1 (0.47) HSD11B1TET3KMT2AFBXL19CXXC5
SCHEMBL1921194 0.71 CHRNB2 (0.47) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL1921191 0.71 CHRNB2 (0.47) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0034415-B1 1-(CYCLOHEXYL OR CYCLOHEXENYL)-4-ARYL-4-PIPERIDINECARBOXYLIC ACID DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1984-05-30 EP disclosed
US-4369184-A ANTIHISTAMINES; HETEROCYCLIC NITRILES JANSSEN PHARMACEUTICA N.V. (BE) 1983-01-18 US disclosed
EP-0034415-A1 1-(Cyclohexyl or cyclohexenyl)-4-aryl-4-piperidinecarboxylic acid derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1981-08-26 EP disclosed