SCHEMBL11119655

SCHEMBL11119655

O=C(O)CCC(=O)C(Cc1ccccc1)NC(=O)OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.61
TACR1 P25103 2/20 0.61
CTSL P07711 2/20 0.60
CTSB P07858 2/20 0.60
CTSS P25774 2/20 0.60
CTSK P43235 2/20 0.60
ALDH1A1 P00352 1/20 0.58
ALOX15 P16050 1/20 0.58
CTRB1 P17538 2/20 0.57
CASP1 P29466 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11119660 1.00 ACE (0.61) ACETACR1CTSLCTSBCTSS
SCHEMBL11119658 1.00 ACE (0.61) ACETACR1CTSLCTSBCTSS
SCHEMBL28356104 0.89 TACR1 (0.64) TACR1CTSLCTSBCTSSCTSK
SCHEMBL11275140 0.88 ALDH1A1 (0.61) ACETACR1CTSLCTSBCTSS
SCHEMBL6330507 0.84 TACR1 (0.62) TACR1CTSLCTSBCTSSCTSK
SCHEMBL13998432 0.84 CTSL (0.64) TACR1CTSLCTSBCTSSCTSK
SCHEMBL4980616 0.84 TACR1 (0.62) ACETACR1CTSLCTSBCTSS
SCHEMBL7327386 0.84 TACR1 (0.62) TACR1CTSLCTSBCTSSCTSK
SCHEMBL6439753 0.84 TACR1 (0.62) ACETACR1CTSLCTSBCTSS
SCHEMBL7490981 0.84 TACR1 (0.62) ACETACR1CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0045161-B1 AMIDES OF 4-OXO-5-AMIDOHEXANOIC ACID DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-03-14 EP disclosed
US-4329473-A HYPOTENSIVE AGENTS SRI INTERNATIONAL 1982-05-11 US disclosed
EP-0045161-A1 Amides of 4-oxo-5-amidohexanoic acid derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-02-03 EP disclosed