SCHEMBL11166554

SCHEMBL11166554

COc1cc(Cc2c(N)nc(N)nc2Cl)cc(OC)c1SC

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.44
ALDH1A1 P00352 1/20 0.43
CYP2D6 P10635 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10678576 0.86 NPSR1 (0.48) NPSR1ALDH1A1CYP2D6ATM
SCHEMBL11821666 0.85 DHFR (0.57) ALDH1A1
SCHEMBL11166121 0.84 ALDH1A1 (0.43) ALDH1A1CYP2D6ATM
SCHEMBL11831045 0.81 DHFR (0.58) NPSR1ALDH1A1CYP2D6ATM
SCHEMBL11859276 0.80 DHFR (0.46) NPSR1ALDH1A1CYP2D6ATM
SCHEMBL11352309 0.80 NPSR1 (0.42) NPSR1ALDH1A1CYP2D6ATM
SCHEMBL12496384 0.77 HSP90AA1 (0.54) NPSR1ALDH1A1
Metioprim SCHEMBL193012 0.75 DHFR (0.73) ALDH1A1
Metioprim SCHEMBL30659007 0.75 DHFR (0.73) ALDH1A1
SCHEMBL11548085 0.73 DHFR (0.65) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0032395-B1 BENZYLPYRIMIDINES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-03-23 EP claimed
EP-0032395-A1 Benzylpyrimidines F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-07-22 EP claimed
EP-0032395-B1 BENZYLPYRIMIDINES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-03-23 EP disclosed
EP-0003212-B1 2.4-DIAMINO-5-BENZYLPYRIMIDINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR PREPARATION F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-03-17 EP disclosed
EP-0032395-A1 Benzylpyrimidines F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-07-22 EP disclosed
EP-0003212-A1 2.4-Diamino-5-benzylpyrimidines, pharmaceutical compositions containing them and their preparation F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1979-08-08 EP disclosed