Metioprim

Metioprim

SCHEMBL193012

COc1cc(Cc2cnc(N)nc2N)cc(OC)c1SC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.73
MEN1 O00255 1/20 0.73
SLC22A1 O15245 1/20 0.73
ALDH1A1 P00352 1/20 0.73
CYP3A4 P08684 1/20 0.73
TSHR P16473 1/20 0.73
NFKB1 P19838 1/20 0.73
CYP2C19 P33261 1/20 0.73
BLM P54132 1/20 0.73
KMT2A Q03164 1/20 0.73
HSD17B10 Q99714 1/20 0.73
HTT P42858 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metioprim SCHEMBL30659007 1.00 DHFR (0.73) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL11548085 0.91 DHFR (0.65) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL11544522 0.91 DHFR (0.65) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL11260435 0.87 DHFR (0.70) DHFRMEN1SLC22A1ALDH1A1CYP3A4
Aditeren SCHEMBL1230789 0.86 DHFR (0.81) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL11257800 0.85 SMN1; SMN2 (0.64) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL9284945 0.85 DHFR (0.79) DHFRMEN1SLC22A1ALDH1A1CYP3A4
Trimethoprim SCHEMBL2637561 0.85 DHFR (1.00) DHFRMEN1SLC22A1ALDH1A1CYP3A4
Trimethoprim SCHEMBL24506 0.85 DHFR (1.00) DHFRMEN1SLC22A1ALDH1A1CYP3A4
Aditeren SCHEMBL10676774 0.85 DHFR (0.79) DHFRMEN1SLC22A1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1167 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4536217-A1 CO-AGENTS AS THERAPY AGAINST ANAEROBIC PATHOGENS Fleurir Abx LLC (US) 2025-04-16 EP claimed
US-20240293434-A1 COMBINATION THERAPY EFFECTIVE AGAINST MICROORGANISMS, INCLUDING DRUG RESISTANT MICROORGANISMS FLEURIR ABX LLC (US) 2024-09-05 US claimed
WO-2023239822-A1 CO-AGENTS AS THERAPY AGAINST ANAEROBIC PATHOGENS FLEURIR ABX LLC (US) 2023-12-14 WO claimed
US-20230398101-A1 Co-agents as Therapy Against Anaerobic Pathogens FLEURIR ABX LLC (US) 2023-12-14 US claimed
US-20220169680-A1 CELL-PENETRATING PEPTIDE BASED ON INFLUENZA VIRUS M2 PROTEIN INSTITUTE OF BASIC MEDICAL SCIENCES CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2022-06-02 US claimed
EP-3923953-A2 PYRIMIDINE DERIVATIVE CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2021-12-22 EP claimed
EP-3912989-A1 CELL-PENETRATING PEPTIDE BASED ON INFLUENZA VIRUS M2 PROTEIN Institute of Basic Medical Sciences Chinese Academy of Medical Sciences (CN) 2021-11-24 EP claimed
WO-2020168358-A2 PYRIMIDINE DERIVATIVE CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2020-08-20 WO claimed
US-20200253994-A1 PYRIMIDINE DERIVATIVE CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2020-08-13 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
EP-1578434-A2 METHODS AND COMPOSITIONS RELATING TO ISOLEUCINE BOROPROLINE COMPOUNDS Point Therapeutics, Inc. (US) 2005-09-28 EP claimed
US-20040131628-A1 Nucleic acids for the treatment of disorders associated with microorganisms BRATZLER ROBERT L (US) 2004-07-08 US claimed
US-20040077601-A1 Methods and compositions relating to isoleucine boroproline compounds POINT THERAPEUTICS, INC. 2004-04-22 US claimed
WO-2004004658-A2 METHODS AND COMPOSITIONS RELATING TO ISOLEUCINE BOROPROLINE COMPOUNDS POINT THERAPEUTICS, INC. (US) 2004-01-15 WO claimed
US-4599416-A Process for the preparation of aqueous solutions of potentiated sulfonamides HOFFMANN-LA ROCHE INC. (US) 1986-07-08 US claimed
EP-0037501-B1 PHARMACEUTICAL PREPARATIONS AND MANUFACATURE F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1984-07-18 EP claimed
EP-0003212-B1 2.4-DIAMINO-5-BENZYLPYRIMIDINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR PREPARATION F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-03-17 EP claimed
EP-0037501-A1 Pharmaceutical preparations and manufacature F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-10-14 EP claimed
US-4180578-A 2,4-Diamino-5-(4'-methylthio)benzylpyrimidenes, compounds, compositions and method of use Ludwig Heumann, & Co. GmbH (DE) 1979-12-25 US claimed
EP-0003212-A1 2.4-Diamino-5-benzylpyrimidines, pharmaceutical compositions containing them and their preparation F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1979-08-08 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240293434-A1 COMBINATION THERAPY EFFECTIVE AGAINST MICROORGANISMS, INCLUDING DRUG RESISTANT MICROORGANISMS SLC11A2, MYD88, FPR2 DHFR 7/4885MEN1 957/4885SLC22A1 3025/4885
US-20040077601-A1 Methods and compositions relating to isoleucine boroproline compounds BCAT1, BCAT2, APOB DHFR 69/4885MEN1 1014/4885SLC22A1 1246/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.