SCHEMBL11187565

SCHEMBL11187565

Cc1cc(C)c(NC2=NCCN2)c(C)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 5/20 0.76
HTR1B P28222 4/20 0.76
CFB P00751 5/20 0.58
ADRA2C P18825 8/20 0.55
ADRA1A P35348 5/20 0.55
KCNH2 Q12809 1/20 0.55
ADRA2A P08913 7/20 0.54
ADRA2B P18089 7/20 0.54
ADRA1D P25100 4/20 0.54
ADRA1B P35368 4/20 0.54
CYP2D6 P10635 2/20 0.53
NISCH Q9Y2I1 2/20 0.53
CYP1A2 P05177 1/20 0.53
TSHR P16473 1/20 0.53
NFKB1 P19838 1/20 0.53
HSD17B10 Q99714 1/20 0.53
LMNA P02545 3/20 0.51
MEN1 O00255 1/20 0.51
SLC22A1 O15245 1/20 0.51
SLC22A3 O75751 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10979251 0.86 HTR1D (0.71) HTR1DHTR1BCFBADRA2CADRA1A
Hydrochloric Acid SCHEMBL10973842 0.85 HTR1D (0.69) HTR1DHTR1BCFBADRA2CADRA1A
SCHEMBL24658874 0.83 ADRA2A (0.71) HTR1DHTR1BCFBADRA2CADRA1A
SCHEMBL4760243 0.82 HTR1D (1.00) HTR1DHTR1BCFBADRA2CADRA1A
Hydrochloric Acid SCHEMBL29384552 0.81 HTR1D (0.97) HTR1DHTR1BCFBADRA2CADRA1A
SCHEMBL6054534 0.77 HTR1D (0.58) HTR1DHTR1BCFBADRA2CADRA1A
SCHEMBL14976356 0.74 CFB (0.67) HTR1DHTR1BCFBADRA2CADRA1A
SCHEMBL8693621 0.74 CFB (0.57) HTR1DHTR1BCFBADRA2CADRA1A
SCHEMBL6054523 0.74 ADRA2A (0.63) HTR1DHTR1BCFBADRA2CADRA1A
SCHEMBL6585037 0.74 HTR1D (0.55) HTR1DHTR1BCFBADRA2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016105449-A1 COMPOUNDS FOR USE AS PAIN THERAPEUTICS LEDERMAN SETH (US) 2016-06-30 WO disclosed
US-4389403-A HYPOTENSIVE AGENTS BASF AKTIENGESELLSCHAFT (DE) 1983-06-21 US disclosed