SCHEMBL1119616

SCHEMBL1119616

CC(=O)Cc1ccc(NC2CCCN(c3nc(-c4ccc(Cl)cc4Cl)cc4nc(C5CCN(C6CC6)CC5)nn34)C2)nc1N

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.38
BTK Q06187 3/20 0.32
JAK3 P52333 3/20 0.32
CCR4 P51679 1/20 0.31
DPP4 P27487 3/20 0.30
IL1B P01584 1/20 0.30
NLRP3 Q96P20 1/20 0.30
F10 P00742 1/20 0.30
CXCR3 P49682 1/20 0.30
CNR1 P21554 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
EGFR P00533 1/20 0.30
LCK P06239 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1962806 0.89 GSK3B (0.38) GSK3BBTKJAK3DPP4CNR1
SCHEMBL8003442 0.81 GSK3B (0.37) GSK3BBTKJAK3CCR4DPP4
SCHEMBL1962175 0.81 GSK3B (0.35) GSK3BBTKJAK3DPP4IL1B
SCHEMBL1119579 0.80 BMPR1B (0.32) BTKJAK3DPP4EGFRLCK
SCHEMBL1120117 0.76 MAPK14 (0.32) GSK3BBTKJAK3IL1BEGFR
SCHEMBL1120237 0.72 GSK3B (0.34) GSK3B
SCHEMBL1962515 0.72 DPP4 (0.34) GSK3BDPP4
SCHEMBL8006538 0.71 GSK3B (0.34) GSK3BDPP4HTTSMN1; SMN2
SCHEMBL16456992 0.71 WNT1 (0.31) BTKJAK3IL1BEGFRLCK
SCHEMBL1120012 0.70 LMNA (0.36) DPP4CNR1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2280976-A1 SUBSTITUTED IMIDAZO- AND TRIAZOLOPYRIMIDINES, IMIDAZO- AND PYRAZOLOPYRAZINES AND IMIDAZOTRIAZINES AS GSK3BETA-INHIBITORS Bayer Schering Pharma Aktiengesellschaft (DE) 2011-02-09 EP disclosed
WO-2009138176-A1 SUBSTITUTED IMIDAZO- AND TRIAZOLOPYRIMIDINES, IMIDAZO- AND PYRAZOLOPYRAZINES AND IMIDAZOTRIAZINES AS GSK3BETA-INHIBITORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-11-19 WO disclosed