SCHEMBL11200372

SCHEMBL11200372

CC(C)(C)OC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN)NC(=O)OCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.60
DPP8 Q6V1X1 3/20 0.60
DPP7 Q9UHL4 2/20 0.56
ADORA3 P0DMS8 1/20 0.54
ADORA2A P29274 1/20 0.54
ADORA2B P29275 1/20 0.54
ADORA1 P30542 1/20 0.54
ITGB3 P05106 1/20 0.51
ITGA2B P08514 1/20 0.51
ACE P12821 4/20 0.49
PRSS8 Q16651 1/20 0.49
F2 P00734 1/20 0.49
PRSS1 P07477 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP3A4 P08684 1/20 0.49
TSHR P16473 1/20 0.49
PREP P48147 2/20 0.47
KLK5 Q9Y337 1/20 0.47
FKBP1A P62942 1/20 0.47
CMA1 P23946 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7321218 0.88 ACE (0.60) ADORA3ADORA2AADORA2BADORA1ACE
SCHEMBL7326774 0.88 DPP8 (0.70) DPP4DPP8DPP7ACEPRSS8
SCHEMBL9040522 0.88 DPP4 (0.67) DPP4DPP8DPP7ACEPREP
SCHEMBL9040510 0.88 DPP4 (0.67) DPP4DPP8DPP7ACEPREP
SCHEMBL10619564 0.88 ITGB3 (0.63) DPP4DPP8DPP7ADORA3ADORA2A
SCHEMBL5971737 0.87 ITGB3 (0.66) DPP4DPP8DPP7ADORA3ADORA2A
SCHEMBL14673535 0.86 ADORA3 (0.54) DPP4DPP8ADORA3ADORA2AADORA2B
SCHEMBL20958585 0.86 ADORA3 (0.54) DPP4DPP8ADORA3ADORA2AADORA2B
SCHEMBL14673533 0.86 ADORA3 (0.54) DPP4DPP8ADORA3ADORA2AADORA2B
SCHEMBL14673534 0.86 ADORA3 (0.54) DPP4DPP8ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0083923-A2 Aminoacyl-containing dipeptide derivatives useful as antihypertensives MERCK & CO. INC. (US) 1983-07-20 EP disclosed