SCHEMBL1120137

SCHEMBL1120137

Cc1ccccc1S(=O)(=O)C=CC#N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.54
TDP1 Q9NUW8 5/20 0.54
MAPT P10636 4/20 0.54
HPGD P15428 4/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
TP53 P04637 3/20 0.54
NPC1 O15118 2/20 0.54
NFKB1 P19838 2/20 0.54
RAB9A P51151 2/20 0.54
CYP1A2 P05177 2/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2D6 P10635 2/20 0.54
CYP2C9 P11712 2/20 0.54
MAPK1 P28482 2/20 0.54
CYP2C19 P33261 2/20 0.54
HSD17B10 Q99714 2/20 0.54
S100A4 P26447 1/20 0.54
MTOR P42345 1/20 0.54
NFKB2 Q00653 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28938489 1.00 ALDH1A1 (0.54) ALDH1A1TDP1MAPTHPGDMEN1
SCHEMBL29634902 0.79 ALDH1A1 (0.60) ALDH1A1TDP1MAPTHPGDMEN1
SCHEMBL20774482 0.79 ALDH1A1 (0.60) ALDH1A1TDP1MAPTHPGDMEN1
SCHEMBL20774483 0.79 ALDH1A1 (0.60) ALDH1A1TDP1MAPTHPGDMEN1
SCHEMBL11834947 0.79 ALDH1A1 (0.55) ALDH1A1TDP1MAPTHPGDMEN1
SCHEMBL11834941 0.79 ALDH1A1 (0.55) ALDH1A1TDP1MAPTHPGDMEN1
SCHEMBL10589798 0.76 HPGD (0.55) ALDH1A1TDP1MAPTHPGDMEN1
SCHEMBL10954580 0.76 ALDH1A1 (0.38) ALDH1A1TDP1TP53KDM4ETSHR
SCHEMBL11835667 0.73 PTGES2 (0.48) ALDH1A1TDP1MAPTHPGDMEN1
SCHEMBL742012 0.73 ALDH1A1 (0.67) ALDH1A1TDP1MAPTHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011130395-A1 INHIBITORS OF FLIP TO TREAT CANCER UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2011-10-20 WO disclosed
US-20110251135-A1 INHIBITORS OF PERITONEAL SEEDING OF CANCER CELLS UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2011-10-13 US disclosed
US-7989495-B2 3-Sulfonyl propenenitriles, e.g., BAY 11-7085 (3-(t-butylphenylsulfonyl)-2-propenenitrile; promoting apoptosis and inhibiting readhesion of cancer cells; antimetastasis agents, particularly for hepatic, parietal or peritoneal area; inhibiting tumorigenesis; antiproliferative agents (not for myeloma) UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2011-08-02 US disclosed
EP-2281077-A2 INHIBITORS OF PERITONEAL SEEDING OF CANCER CELLS University of Utah Research Foundation (US) 2011-02-09 EP disclosed
WO-2009124272-A2 INHIBITORS OF PERITONEAL SEEDING OF CANCER CELLS UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2009-10-08 WO disclosed
US-20050124590-A1 Compositions and methods for inhibiting nf-kappab mediated tumorigenicity and adhesion dependent survival of cancer cells NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2005-06-09 US disclosed
WO-2003072038-A2 COMPOSITIONS AND METHODS FOR INHIBITING NF-κB MEDIATED TUMORIGENICITY AND ADHESION-DEPENDENT SURVIVAL OF CANCER CELLS UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2003-09-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050124590-A1 Compositions and methods for inhibiting nf-kappab mediated tumorigenicity and adhesion dependent survival of cancer cells NFKBIA, RELA, NFKB1 ALDH1A1 1727/4885TDP1 2499/4885MAPT 4444/4885
US-20110251135-A1 INHIBITORS OF PERITONEAL SEEDING OF CANCER CELLS NFKBIA, IKBKB, RELA ALDH1A1 2392/4885TDP1 3746/4885MAPT 3675/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.