Bromide

Bromide

SCHEMBL11203752

Br.Oc1cccc(C2=CCCNC2)c1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA2A known ✓ P08913 1/20 0.53
ADRA2B known ✓ P18089 1/20 0.53
HTR2A P28223 5/20 0.43
HSD17B1 P14061 9/20 0.42
HSD17B2 P37059 8/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
ESR1 P03372 2/20 0.37
ESR2 Q92731 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
PIK3CD O00329 1/20 0.36
METAP2 P50579 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11199688 0.98 ADRA2A (0.54) ADRA2AADRA2BHTR2AHSD17B1HSD17B2
SCHEMBL10354111 0.81 HSD17B1 (0.47) HSD17B1HSD17B2CYP3A4CYP2C9HTR2C
Hydrochloric Acid SCHEMBL11019773 0.79 PIK3CD (0.46) HSD17B1HSD17B2CYP3A4CYP2C9HTR2C
Bromide SCHEMBL11196323 0.78 ADRA2A (0.58) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL14904833 0.78 ADRA2A (0.54) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL9311684 0.78 ADRA2A (0.54) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL13490468 0.78 ADRA2A (0.54) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL8959992 0.78 HTR2C (0.57) ADRA2AADRA2BHTR2ACYP3A4CYP2C9
SCHEMBL8960049 0.77 ADRA2A (0.61) ADRA2AADRA2BHTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL9310385 0.77 ADRA2A (0.53) ADRA2AADRA2BHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4382942-A ANTIEMETICS, PARKINSON*S DISEASE ROUSSEL UCLAF (FR) 1983-05-10 US disclosed