SCHEMBL8960049

SCHEMBL8960049

Oc1ccc(C2=CCCNC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.61
ADRA2B P18089 1/20 0.61
QDPR P09417 2/20 0.53
HTR2A P28223 5/20 0.39
HTR2C P28335 2/20 0.39
HTR2B P41595 2/20 0.39
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
TSHR P16473 1/20 0.38
SLC6A1 P30531 1/20 0.38
SLC6A13 Q9NSD5 1/20 0.38
CHRM2 P08172 2/20 0.38
CHRM3 P20309 1/20 0.38
BLM P54132 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29140051 0.80 ADRA2A (0.61) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL8960144 0.80 ADRA2A (0.61) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL8960083 0.80 ADRA2A (0.61) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL10354311 0.79 QDPR (0.68) ADRA2AADRA2BQDPRHTR2CESR1
SCHEMBL4789087 0.79 ADRA2A (0.59) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL13490583 0.79 CHRM2 (0.43) ADRA2AADRA2BQDPRHTR2AHTR2C
Bromide SCHEMBL11196323 0.78 ADRA2A (0.58) ADRA2AADRA2BQDPRHTR2AHTR2C
Hydrochloric Acid SCHEMBL10354312 0.78 QDPR (0.66) ADRA2AADRA2BQDPRHTR2CESR1
Hydrochloric Acid SCHEMBL9252509 0.78 ADRA2A (0.58) ADRA2AADRA2BHTR2AHTR2CHTR2B
SCHEMBL29140044 0.77 ADRA2A (0.57) ADRA2AADRA2BHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109810047-A (R) synthetic method of the chiral intermediate of -3- Phenylpiperidine or/and (S) -3- Phenylpiperidine and Ni Lapani 上海博邦医药科技有限公司 2019-05-28 CN disclosed
EP-0691956-A1 3-PHENYL-1,2,5,6-TETRAHYDROPYRIDINE DERIVATIVES AS SEDATIVES LABORATOIRE L. LAFON (FR) 1996-01-17 EP disclosed
WO-1994022827-A1 3-PHENYL-1,2,5,6-TETRAHYDROPYRIDINE DERIVATIVES AS SEDATIVES LABORATOIRE L. LAFON (FR) 1994-10-13 WO disclosed