SCHEMBL11207304

SCHEMBL11207304

NC(c1ccccc1)C1Sc2ccccc2C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
ADORA3 P0DMS8 1/20 0.37
THRB P10828 1/20 0.37
CHRM1 P11229 1/20 0.37
TBXA2R P21731 1/20 0.37
PTGS1 P23219 1/20 0.37
ADRA1A P35348 1/20 0.37
MAPT P10636 5/20 0.36
MAPK1 P28482 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
TP53 P04637 2/20 0.36
LMNA P02545 1/20 0.36
HTR2B P41595 1/20 0.36
DPP4 P27487 2/20 0.33
F2 P00734 1/20 0.33
TSHR P16473 2/20 0.33
CYP2D6 P10635 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11205372 0.88 TP53 (0.36) KMT2AMEN1PTGS1MAPTMAPK1
SCHEMBL11201233 0.82 ELANE (0.39) KMT2AMEN1MAPTMAPK1CYP1A2
SCHEMBL11413848 0.78
SCHEMBL11200277 0.78 MEN1 (0.33) KMT2AMEN1MAPTNPC1RAB9A
SCHEMBL11211362 0.77 ALDH1A1 (0.44) KMT2AMAPTCYP1A2CYP3A4TP53
SCHEMBL11404541 0.76 EPHX1 (0.40) KMT2AMEN1ADORA3THRBCHRM1
SCHEMBL11402204 0.76 KMT2A (0.34) KMT2AMEN1ADORA3THRBCHRM1
SCHEMBL11204824 0.71 ALDH1A1 (0.36) KMT2AMEN1ADORA3THRBCHRM1
SCHEMBL13940537 0.68 MEN1 (0.41) KMT2AMEN1THRBMAPTMAPK1
SCHEMBL13302892 0.65 ACHE (0.39) KMT2AMEN1THRBMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0091041-A2 Vinylogous carboxamides, process for preparing them and medicines containing these compounds Dr. Karl Thomae GmbH (DE) 1983-10-12 EP disclosed
EP-0025489-A1 Vinylogous carboxamides, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1981-03-25 EP disclosed