SCHEMBL11208796

SCHEMBL11208796

Clc1ccc2c(c1Cl)C=NCC2

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.36
HTR2C P28335 4/20 0.36
HTR2B P41595 3/20 0.36
PNMT P11086 10/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11337914 0.89 PNMT (0.39) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL9573119 0.76 ADRA2A (0.39) HTR2CPNMTADRA2AADRA2BADRA2C
SCHEMBL30908737 0.68 NOTUM (0.46) HTR2AHTR2CHTR2BADRA2AADRA2B
SCHEMBL18524345 0.65
SCHEMBL9573156 0.64 HTR2A (0.38) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL7321373 0.64 HTR2A (0.48) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL9510557 0.64 HTR2A (0.35) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL9573416 0.63 CHRNB2 (0.33)
SCHEMBL184440 0.63 ALK (0.30)
SCHEMBL17372829 0.60 PNMT (0.31) PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0040990-B1 ANTIALLERGIC IMIDODISULFAMIDES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITHKLINE BECKMAN CORPORATION (US) 1983-06-01 EP disclosed
US-4317826-A TREATING ASTHMA SMITHKLINE CORPORATION (US) 1982-03-02 US disclosed
EP-0040990-A1 Antiallergic imidodisulfamides, their preparation and pharmaceutical compositions containing them SMITHKLINE BECKMAN CORPORATION (US) 1981-12-02 EP disclosed