SCHEMBL11213705

SCHEMBL11213705

COc1ncc(CC(C)C)nc1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
PDE10A Q9Y233 2/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
P2RX3 P56373 1/20 0.33
P2RX2 Q9UBL9 1/20 0.33
RORC P51449 2/20 0.32
HTT P42858 1/20 0.31
RECQL P46063 1/20 0.31
S1PR1 P21453 1/20 0.31
ABCB11 O95342 1/20 0.31
PIK3CA P42336 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
HIF1A Q16665 1/20 0.31
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30
PDCD1 Q15116 2/20 0.30
CD274 Q9NZQ7 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16432838 0.86 NOS3 (0.36) NOS3NOS1NOS2PDE10ATRPM8
SCHEMBL30505752 0.85 TRPM8 (0.37) NOS3NOS1NOS2PDE10ATRPM8
SCHEMBL29131679 0.85 TRPM8 (0.37) NOS3NOS1NOS2PDE10ATRPM8
SCHEMBL29070262 0.84 CYP1A2 (0.35) NOS3NOS1NOS2CYP1A2CYP2C9
SCHEMBL29070263 0.82 NOS2 (0.33) NOS2CYP1A2CYP2C9HIF1A
SCHEMBL23131526 0.79 APOBEC3A (0.34) NOS3NOS2PDE10AHTTRECQL
SCHEMBL9953928 0.79 NOS3 (0.41) NOS3NOS1NOS2PDE10ACYP1A2
SCHEMBL31374320 0.79 NOS3 (0.41) NOS3NOS1NOS2PDE10ACYP1A2
SCHEMBL31442989 0.79 TRPM8 (0.38) NOS3NOS1NOS2PDE10ATRPM8
SCHEMBL31442991 0.79 TRPM8 (0.38) NOS3NOS1NOS2PDE10ATRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-57062269-A None JP disclosed
JP-S5762269-A 2,3,5-TRISUBSTITUTED PYRAZINE DERIVATIVE OGAWA KORYO KK 1982-04-15 JP disclosed