SCHEMBL11215917

SCHEMBL11215917

C=CCn1c(=O)[nH]c(=O)c2[nH]c(N)nc21

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.43
PDE4B Q07343 2/20 0.43
PDE4C Q08493 2/20 0.43
PDE4D Q08499 2/20 0.43
PDE5A O76074 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PNP P00491 2/20 0.41
ADORA2B P29275 3/20 0.40
ADORA3 P0DMS8 1/20 0.40
ALDH1A1 P00352 2/20 0.39
ADORA2A P29274 3/20 0.38
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 2/20 0.37
RECQL P46063 1/20 0.37
PKM P14618 1/20 0.37
ADORA1 P30542 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5183524 0.85 PDE5A (0.41) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL4623642 0.82 ALDH1A1 (0.41) MEN1KMT2AADORA2BADORA3ALDH1A1
SCHEMBL18039294 0.82 ADORA2B (0.40) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL8947982 0.81 POLB (0.40) ADORA2BADORA3ALDH1A1ADORA2APOLB
SCHEMBL6755794 0.78 ADORA2B (0.38) ADORA2BADORA3ALDH1A1ADORA2APOLB
SCHEMBL18036533 0.76 ADORA2B (0.38) MEN1KMT2AADORA2BADORA3ALDH1A1
SCHEMBL5134359 0.76 ADORA2A (0.66) PDE4APDE4BPDE4CPDE4DPNP
SCHEMBL11591427 0.76 ADORA2B (0.57) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7345938 0.75 PDE5A (0.66) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL4551932 0.75 TRAP1 (0.54) ADORA2BADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4397779-A RADIOIMMUNOASSAY OF THEOPHYLLINE AND DERIVATIVES; IODINATION BAXTER TRAVENOL LABORATORIES, INC. (US) 1983-08-09 US disclosed
US-4297494-A Xanthine tracers BAXTER TRAVENOL LABORATORIES, INC. (US) 1981-10-27 US disclosed