SCHEMBL11220600

SCHEMBL11220600

CCC1OC2(CCN(CCC3COc4ccccc4O3)CC2)CNC1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.46
OPRM1 P35372 3/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
HIF1A Q16665 1/20 0.43
NR1I2 O75469 1/20 0.43
LMNA P02545 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
DRD4 P21917 1/20 0.43
SLC6A2 P23975 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11235292 0.90 DRD2 (0.44) DRD2OPRM1MEN1CYP1A2CYP3A4
SCHEMBL11236298 0.88 DRD2 (0.47) DRD2OPRM1MEN1CYP1A2CYP3A4
SCHEMBL11224414 0.83 SIGMAR1 (0.62) DRD2OPRM1KCNH2SIGMAR1
SCHEMBL11234750 0.82 DRD2 (0.44) DRD2OPRM1MEN1CYP1A2CYP3A4
SCHEMBL11219845 0.80 DRD2 (0.39) DRD2OPRM1MEN1CYP1A2CYP3A4
SCHEMBL11220552 0.80 DRD2 (0.47) DRD2OPRM1MEN1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11226124 0.79 DRD2 (0.46) DRD2OPRM1MEN1CYP1A2CYP3A4
SCHEMBL11292608 0.77 SIGMAR1 (0.67) OPRM1CYP2D6TSHRKMT2ALMNA
SCHEMBL11234698 0.76 OPRM1 (0.47) DRD2OPRM1KCNH2SIGMAR1
SCHEMBL11224595 0.75 SIGMAR1 (0.61) DRD2OPRM1KCNH2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4353901-A HYPERTENSION, CONGESTIVE HEART FAILURE, ARRHYTHMIAMIGRAINE, VASOSPASTIC DISORDERS, ASTHMA SYNTEX (U.S.A.) INC. (US) 1982-10-12 US disclosed