SCHEMBL11221253

SCHEMBL11221253

CCCCC1OC2(CCN(CC(O)C3COc4ccccc4O3)CC2)C(C)NC1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.35
KMT2A Q03164 3/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
HIF1A Q16665 1/20 0.35
NR1I2 O75469 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
DRD4 P21917 1/20 0.35
SLC6A2 P23975 1/20 0.35
ADRA1D P25100 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11230155 0.91 DRD2 (0.37) DRD2KMT2ALMNAMEN1CYP2D6
SCHEMBL11220765 0.87 DRD2 (0.39) DRD2KMT2ALMNAMEN1CYP2D6
SCHEMBL11238198 0.83 DRD2 (0.42) DRD2KMT2ALMNAMEN1CYP2D6
SCHEMBL11235867 0.81 ALDH1A1 (0.36) DRD2KMT2ALMNAMEN1CYP2D6
Hydrochloric Acid SCHEMBL11371592 0.81 DRD2 (0.39) DRD2KMT2ALMNAMEN1CYP2D6
SCHEMBL11225550 0.80 DRD2 (0.39) DRD2KMT2ALMNAMEN1CYP2D6
SCHEMBL11224661 0.78 OPRM1 (0.41) DRD2KMT2AOPRM1ALDH1A1
SCHEMBL11230804 0.78 LMNA (0.37) DRD2KMT2ALMNAMEN1CYP2D6
SCHEMBL11370777 0.76 ALDH1A1 (0.39) DRD2KMT2ALMNAMEN1CYP2D6
SCHEMBL11219845 0.75 DRD2 (0.39) DRD2KMT2ALMNAMEN1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4353901-A HYPERTENSION, CONGESTIVE HEART FAILURE, ARRHYTHMIAMIGRAINE, VASOSPASTIC DISORDERS, ASTHMA SYNTEX (U.S.A.) INC. (US) 1982-10-12 US disclosed