SCHEMBL11224620

SCHEMBL11224620

COc1ccc2c(c1)CC1CCC(C2)C1=O

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.53
DRD3 P35462 5/20 0.53
CYP19A1 P11511 3/20 0.50
ACHE P22303 5/20 0.49
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
METAP1 P53582 2/20 0.46
CA1 P00915 4/20 0.46
CA2 P00918 4/20 0.46
CYP26A1 O43174 1/20 0.46
DRD4 P21917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11219696 0.81 DRD2 (0.44) DRD2DRD3CYP19A1ACHEMTNR1A
SCHEMBL11225618 0.81 DRD2 (0.44) DRD2DRD3CYP19A1ACHEMTNR1A
SCHEMBL11221031 0.79 DRD2 (0.49) DRD2DRD3CYP19A1ACHEMTNR1A
SCHEMBL11221034 0.79 DRD2 (0.49) DRD2DRD3CYP19A1ACHEMTNR1A
SCHEMBL13241438 0.77 ACHE (0.44) ACHEMETAP1
SCHEMBL13241439 0.77 ACHE (0.44) ACHEMETAP1
SCHEMBL6053239 0.76 CYP19A1 (0.45) CYP19A1
SCHEMBL13866813 0.76 DRD2 (0.50) DRD2DRD3CA1CA2DRD4
SCHEMBL4361668 0.76 ALDH1A1 (0.49) DRD2DRD3CYP19A1MTNR1AMTNR1B
SCHEMBL13799409 0.76 DRD2 (0.56) DRD2DRD3CYP19A1ACHEMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4332810-A N-(Substituted)-2,5-ethano-8-hydroxy (or methoxy)-1,2,3,4,5,6-hexahydro-3 (or 4)-benzazocine centrally-acting analgesics MERCK & CO., INC. (US) 1982-06-01 US disclosed