SCHEMBL6053239

SCHEMBL6053239

O=C1C2CCC1Cc1cc(Oc3ccncc3)ccc1C2

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.45
FAAH O00519 14/20 0.43
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11224620 0.76 DRD2 (0.53) CYP19A1
SCHEMBL13866813 0.71 DRD2 (0.50)
SCHEMBL346240 0.70 FAAH (0.61) CYP19A1FAAH
SCHEMBL346899 0.70 FAAH (0.54) FAAH
SCHEMBL346830 0.70 FAAH (0.49) FAAH
SCHEMBL4045668 0.69 MAOA (0.52) FAAH
SCHEMBL13241438 0.67 ACHE (0.44)
SCHEMBL13866811 0.67 DRD2 (0.49) CYP19A1CYP11B2
SCHEMBL4045125 0.67 PSEN1 (0.42)
SCHEMBL1025843 0.67 DRD2 (0.49) CYP19A1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268412-B1 SULPHONAMIDO-SUBSTITUTED BRIDGED BICYCLOALKYL DERIVATIVES MERCK SHARP & DOHME (GB) 2006-11-22 EP disclosed