SCHEMBL11225248

SCHEMBL11225248

c1ccc(Cc2cc3ccccc3[nH]2)nc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.55
LOXL2 Q9Y4K0 1/20 0.51
AHR P35869 2/20 0.49
HRH3 Q9Y5N1 2/20 0.49
HRH4 Q9H3N8 1/20 0.49
PCSK9 Q8NBP7 3/20 0.46
CYP1A2 P05177 1/20 0.43
CYP2E1 P05181 1/20 0.43
CYP2C8 P10632 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2B6 P20813 1/20 0.43
CYP2C19 P33261 1/20 0.43
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
GUSB P08236 1/20 0.43
F2 P00734 1/20 0.42
F10 P00742 1/20 0.42
F7 P08709 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6616428 0.83 HRH3 (0.43) IDO1LOXL2AHRHRH3HRH4
SCHEMBL28338445 0.80 LOXL2 (0.69) LOXL2AHRHRH3HRH4PCSK9
SCHEMBL401081 0.80 LOXL2 (0.69) LOXL2AHRHRH3HRH4PCSK9
SCHEMBL29403791 0.80 LOXL2 (0.69) LOXL2AHRHRH3HRH4PCSK9
SCHEMBL28335219 0.78 LOXL2 (0.67) LOXL2AHRHRH3PCSK9MTNR1A
SCHEMBL28836433 0.76 AHR (0.49) LOXL2AHRPCSK9GUSB
SCHEMBL10677541 0.75 HRH3 (0.48) IDO1LOXL2AHRHRH3HRH4
SCHEMBL6988526 0.75 LOXL2 (0.53) IDO1LOXL2AHRHRH3HRH4
Pyridine SCHEMBL27581580 0.74 F2 (0.49) IDO1LOXL2AHRF2
SCHEMBL6758056 0.74 TAAR1 (0.51) LOXL2AHRPCSK9GUSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4363912-A 3-PYRIDYL-3-OR-4-ALKYL INDOLES PFIZER INC. (US) 1982-12-14 US disclosed
US-4101583-A Alpha-methylthio-alpha-(2-aminophenyl) acetaldehyde diloweralkyl acetals THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1978-07-18 US disclosed
US-4080341-A Carbazolenine and indole compounds THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1978-03-21 US disclosed
US-4067875-A Certain N-phenyl or N-pyridyl aza sulfonium salts THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1978-01-10 US disclosed
US-3992392-A Synthesis of indoles from anilines and intermediates therein THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1976-11-16 US disclosed