SCHEMBL11233385

SCHEMBL11233385

COc1c(-c2nc3cncnc3[nH]2)ccc(C)c1S

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 5/20 0.41
PDE5A O76074 2/20 0.32
EGFR P00533 2/20 0.31
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11352539 0.88 AMY1A (0.31) AMY1A
SCHEMBL10691368 0.82 AMY1A (0.41) AMY1AALDH1A1CYP3A4
SCHEMBL10960693 0.79 EGFR (0.36) AMY1APDE5AEGFRALDH1A1CYP3A4
SCHEMBL7279881 0.79 AMY1A (0.47) AMY1APDE5AALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL7277923 0.78 AMY1A (0.46) AMY1APDE5AALDH1A1SMN1; SMN2
SCHEMBL10963776 0.76 PDE5A (0.39) AMY1APDE5AALDH1A1CYP3A4HSD17B10
SCHEMBL10962015 0.75 ESR1 (0.36) AMY1AEGFRCYP3A4
SCHEMBL10965568 0.75 METAP2 (0.41) AMY1APDE5AALDH1A1HSD17B10
SCHEMBL10678378 0.75 AMY1A (0.49) AMY1APDE5AALDH1A1SMN1; SMN2HSD17B10
SCHEMBL10961186 0.75 TNKS (0.33) AMY1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024290-B1 8-PHENYL PURINES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1982-12-22 EP claimed
US-4299834-A INOTROPIC ACTIVITY BOEHRINGER INGELHEIM GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-11-10 US claimed
EP-0024290-A1 8-Phenyl purines, their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1981-03-04 EP claimed
EP-0024290-B1 8-PHENYL PURINES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1982-12-22 EP disclosed
US-4299834-A INOTROPIC ACTIVITY BOEHRINGER INGELHEIM GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-11-10 US disclosed
EP-0024290-A1 8-Phenyl purines, their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1981-03-04 EP disclosed