SCHEMBL11235524

SCHEMBL11235524

CC(=O)Nc1nn(C)c2nc(C)c(-c3ccncc3)cc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.56
CASP1 P29466 8/20 0.56
CASP7 P55210 8/20 0.56
HSD17B10 Q99714 8/20 0.56
MAPT P10636 5/20 0.56
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
LMNA P02545 1/20 0.56
PDE3B Q13370 2/20 0.47
PDE3A Q14432 2/20 0.47
ALDH1A1 P00352 6/20 0.46
L3MBTL1 Q9Y468 2/20 0.43
GLA P06280 1/20 0.43
HPGD P15428 2/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NR1I2 O75469 2/20 0.42
AHR P35869 2/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11229128 0.85 KDM4E (0.50) KDM4ECASP1CASP7HSD17B10MAPT
SCHEMBL11240415 0.82 KMT2A (0.46) KDM4ECASP1CASP7HSD17B10MAPT
SCHEMBL11223425 0.81 PDE3B (0.46) KDM4ECASP1CASP7HSD17B10MAPT
SCHEMBL11231889 0.78 KDM4E (0.49) KDM4ECASP1CASP7HSD17B10MAPT
SCHEMBL11232990 0.76 PDE3B (0.51) HSD17B10PDE3BPDE3AALDH1A1HPGD
SCHEMBL11225855 0.74 PDE3B (0.49) HSD17B10PDE3BPDE3AALDH1A1HPGD
SCHEMBL18604300 0.72 PDE3B (0.43) KDM4EPDE3BPDE3AALDH1A1HPGD
SCHEMBL11233210 0.69 MEN1 (0.43) KDM4ECASP1CASP7HSD17B10MAPT
SCHEMBL11235962 0.68 PDE3B (0.42) KDM4ECASP1CASP7HSD17B10MAPT
SCHEMBL11238184 0.68 MAPK10 (0.43) KDM4ECASP1CASP7HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4361568-A 5-(Pyridinyl)-1H-pyrazolo[3,4-b]pyridin-3-amines and their cardiotonic use STERLING DRUG INC. (US) 1982-11-30 US disclosed
EP-0063754-A1 Pyrazolopyridine derivatives, and preparation, useful as cardiotonics STERLING DRUG INC. (US) 1982-11-03 EP disclosed
EP-0058505-A1 Preparation of esters containing an alpha-cyano group in the alcohol portion of the esters FMC Corporation (US) 1982-08-25 EP disclosed