SCHEMBL11236002

SCHEMBL11236002

CC(=O)SCC(CC(C)C)C(=O)NCC(=O)NCCCCNC(=N)N

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ABCC3 O15438 1/20 0.33
NR1I2 O75469 1/20 0.33
ABCB11 O95342 1/20 0.33
NR3C1 P04150 1/20 0.33
RARG P13631 1/20 0.33
CNR1 P21554 1/20 0.33
OPRK1 P41145 1/20 0.33
NR1H2 P55055 1/20 0.33
PPARA Q07869 1/20 0.33
NR1H3 Q13133 1/20 0.33
NR1I3 Q14994 1/20 0.33
KISS1R Q969F8 1/20 0.33
NPY4R P50391 9/20 0.32
NPY5R Q15761 9/20 0.32
NPY1R P25929 8/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11268857 0.91 KISS1R (0.37) CYP1A2CYP3A4CYP2C19KISS1RNPY4R
SCHEMBL10919519 0.86 NPY4R (0.44) NPY4RNPY5RNPY1RNPY2RFCER2
SCHEMBL10919416 0.86 NPY4R (0.39) OPRK1NPY4RNPY5RNPY1RNPY2R
SCHEMBL9068526 0.85 NPY4R (0.40) NPY4RNPY5RNPY1RNPY2RMME
SCHEMBL10916522 0.83 CYP1A2 (0.37) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL10914759 0.83 NPY4R (0.34) CYP1A2KISS1RNPY4RNPY5RNPY1R
SCHEMBL10918462 0.82 NPY4R (0.44) OPRK1NPY4RNPY5RNPY1RNPY2R
SCHEMBL11207356 0.79 NPY4R (0.46) NPY4RNPY5RNPY1RNPY2R
SCHEMBL10922325 0.79 CYP1A2 (0.35) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11209304 0.79 MMP8 (0.39) CYP3A4CYP2C19KISS1RMMECPB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0067429-A1 Inhibitors of mammalian collagenase E.R. Squibb & Sons, Inc. (US) 1982-12-22 EP disclosed