SCHEMBL11236724

SCHEMBL11236724

CCCCCc1nc(Cl)c(Cl)cc1-c1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.38
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 1/20 0.37
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
GCGR P47871 4/20 0.36
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
NFKB1 P19838 1/20 0.35
S1PR1 P21453 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GRM2 Q14416 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11236919 0.95 GSK3B (0.42) GSK3BCYP3A4CYP2D6PDE3BPDE3A
SCHEMBL11235206 0.91 PDE3B (0.38) GSK3BCYP3A4CYP2D6PDE3BPDE3A
SCHEMBL7278975 0.84 PDE3B (0.49) GSK3BPDE3BPDE3AALDH1A1NPC1
SCHEMBL11247476 0.82 PDE3B (0.36) GSK3BCYP3A4CYP2D6PDE3BPDE3A
SCHEMBL11245026 0.82 PDE3B (0.48) GSK3BCYP3A4PDE3BPDE3AALDH1A1
SCHEMBL11248447 0.81 SMN1; SMN2 (0.40) GSK3BCYP3A4CYP2D6PDE3BPDE3A
SCHEMBL11156699 0.80 CASP1 (0.47) MAPTCNR1
SCHEMBL11176428 0.79 CYP3A4 (0.39) GSK3BCYP3A4CYP2D6GCGRALDH1A1
SCHEMBL11381156 0.79 CYP46A1 (0.47) CNR1CNR2
SCHEMBL11242799 0.78 PDE3B (0.49) GSK3BPDE3BPDE3AGCGRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4351941-A Pyridinyl-pyridines STERLING DRUG INC. (US) 1982-09-28 US disclosed
US-4331672-A 5-(Pyridinyl)pyridine-2-hydrazines, their preparation and their cardiotonic use STERLING DRUG INC. (US) 1982-05-25 US disclosed