SCHEMBL11248447

SCHEMBL11248447

CCCCc1nc(Cl)c(Br)cc1-c1ccncc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.40
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 2/20 0.40
NFKB1 P19838 2/20 0.40
RAB9A P51151 2/20 0.40
NFKB2 Q00653 2/20 0.40
RELA Q04206 2/20 0.40
GSK3B P49841 1/20 0.40
MAPT P10636 1/20 0.40
S1PR1 P21453 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GCGR P47871 6/20 0.38
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
LATS1 O95835 2/20 0.33
MAPK1 P28482 2/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
MAPK14 Q16539 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11236919 0.85 GSK3B (0.42) SMN1; SMN2ALDH1A1NPC1NFKB1RAB9A
SCHEMBL11236724 0.81 GSK3B (0.38) SMN1; SMN2ALDH1A1NPC1NFKB1RAB9A
SCHEMBL11242799 0.80 PDE3B (0.49) SMN1; SMN2ALDH1A1NPC1NFKB1RAB9A
SCHEMBL11235206 0.78 PDE3B (0.38) ALDH1A1NPC1RAB9AGSK3BMAPT
SCHEMBL11156606 0.78 CASP1 (0.48) GSK3BMAPT
SCHEMBL11237097 0.78 POLB (0.41) SMN1; SMN2ALDH1A1NPC1NFKB1RAB9A
SCHEMBL7280225 0.76 MAPT (0.40) SMN1; SMN2ALDH1A1NPC1NFKB1RAB9A
SCHEMBL11245026 0.76 PDE3B (0.48) ALDH1A1GSK3BNPSR1CYP3A4PDE3B
SCHEMBL11394299 0.76 CYP46A1 (0.48) GSK3B
SCHEMBL7272903 0.75 PDE3B (0.44) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4351941-A Pyridinyl-pyridines STERLING DRUG INC. (US) 1982-09-28 US disclosed
US-4331672-A 5-(Pyridinyl)pyridine-2-hydrazines, their preparation and their cardiotonic use STERLING DRUG INC. (US) 1982-05-25 US disclosed