SCHEMBL11238864

SCHEMBL11238864

CC(C)Cc1nc2c(cc1-c1ccncc1)c(N)nn2CCO

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.36
MAPK1 P28482 2/20 0.36
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34
MAP4K1 Q92918 2/20 0.33
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
GSK3B P49841 1/20 0.32
KCNH2 Q12809 1/20 0.32
DYRK1A Q13627 1/20 0.32
BRAF P15056 3/20 0.31
ABL1 P00519 3/20 0.31
BMPR1B O00238 2/20 0.31
CIT O14578 2/20 0.31
RIPK2 O43353 2/20 0.31
STK10 O94804 2/20 0.31
MAP4K4 O95819 2/20 0.31
RAF1 P04049 2/20 0.31
ERBB3 P21860 2/20 0.31
JAK1 P23458 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11245015 0.87 PDE3B (0.39) AAK1MAPK1AKT1AKT2MAP4K1
SCHEMBL11240784 0.82 PDE3B (0.46) MAPK1AKT1AKT2MAP4K1ROCK2
SCHEMBL11231193 0.77 MAPK1 (0.39) MAPK1AKT1AKT2GSK3B
SCHEMBL11382554 0.77 GSK3B (0.38) AAK1ROCK2GSK3BKCNH2DYRK1A
SCHEMBL11244896 0.72 GSK3B (0.49) MAPK1AKT1ROCK2ROCK1GSK3B
SCHEMBL11238221 0.72 PDE3B (0.41) AAK1MAPK1AKT1AKT2GSK3B
SCHEMBL11227748 0.71 MAPT (0.39) AAK1MAPK1AKT1AKT2ROCK2
SCHEMBL11165444 0.70 GSK3B (0.40) AAK1GSK3BPDE3BPDE3A
SCHEMBL11246839 0.70 GSK3B (0.38) MAPK1AKT1AKT2ROCK2GSK3B
SCHEMBL11367530 0.70 PDE3B (0.40) MAPK1BRAFMAPK3JAK2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4361568-A 5-(Pyridinyl)-1H-pyrazolo[3,4-b]pyridin-3-amines and their cardiotonic use STERLING DRUG INC. (US) 1982-11-30 US disclosed
US-4264603-A 5-(Pyridinyl)-1H-pyrazolo[3,4-b]pyridine-3-amines, their use as cardiotonics and their preparation STERLING DRUG INC. (US) 1981-04-28 US disclosed