SCHEMBL11239680

SCHEMBL11239680

O=C(O)C1(c2ccccc2Oc2ccc(F)cc2)CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 8/20 0.46
SLC6A4 P31645 8/20 0.46
SLC6A3 Q01959 8/20 0.46
HTR1A P08908 6/20 0.46
SIGMAR1 Q99720 1/20 0.40
OPRM1 P35372 1/20 0.39
SCN8A Q9UQD0 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
MAP2K1 Q02750 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PARP10 Q53GL7 1/20 0.37
REN P00797 1/20 0.36
EGFR P00533 1/20 0.36
MMP3 P08254 1/20 0.36
MMP10 P09238 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL11471759 0.99 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3HTR1ASIGMAR1
SCHEMBL11248093 0.92 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3HTR1ASIGMAR1
Bromide SCHEMBL11470442 0.91 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3HTR1ASIGMAR1
SCHEMBL11239682 0.82 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3HTR1ASIGMAR1
SCHEMBL11255002 0.82 OPRM1 (0.45) SLC6A2SLC6A4SLC6A3HTR1ASIGMAR1
SCHEMBL5498370 0.81 CTNNB1 (0.46) ALDH1A1MAPTLMNAL3MBTL1
SCHEMBL11477208 0.81 SIGMAR1 (0.44) SLC6A2SLC6A4SLC6A3HTR1ASIGMAR1
Bromide SCHEMBL11242341 0.81 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3HTR1ASIGMAR1
SCHEMBL11241289 0.80 KMT2A (0.44) ALDH1A1MAPK1
SCHEMBL11476866 0.78 OPRM1 (0.47) SLC6A2SLC6A4SLC6A3HTR1ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4198417-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US claimed
EP-0016261-B1 SPIRO(DIBENZ(B,F)OXEPIN-PIPERIDINES) AND METHODS OF PREPARING SAME HOECHST AKTIENGESELLSCHAFT (DE) 1982-12-29 EP disclosed
US-4198417-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed
US-4198418-A ANALGESICS, TRANQUILIZERS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed