SCHEMBL11241289

SCHEMBL11241289

CC(=O)N1CCC(C(=O)O)(c2ccccc2Oc2ccc(F)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
RAB9A P51151 1/20 0.44
USP2 O75604 2/20 0.41
ALDH1A1 P00352 4/20 0.40
CYP2C19 P33261 3/20 0.40
MAPK1 P28482 2/20 0.40
S1PR2 O95136 3/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
CYP2D6 P10635 4/20 0.40
TSHR P16473 1/20 0.40
CYP3A4 P08684 3/20 0.39
CYP2C9 P11712 2/20 0.39
CYP1A2 P05177 1/20 0.38
HPGD P15428 1/20 0.38
ALOX12 P18054 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TET3 O43151 1/20 0.38
FBXL19 Q6PCT2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11242994 0.93 USP2 (0.45) KMT2AMEN1RAB9AUSP2ALDH1A1
SCHEMBL11255002 0.88 OPRM1 (0.45) ALDH1A1
SCHEMBL11471965 0.85 MEN1 (0.43) KMT2AMEN1RAB9AUSP2ALDH1A1
SCHEMBL11486442 0.85 USP2 (0.45) KMT2AMEN1RAB9AUSP2ALDH1A1
SCHEMBL11241295 0.84 USP2 (0.40) KMT2AMEN1RAB9AUSP2ALDH1A1
SCHEMBL11244293 0.83 CYP2D6 (0.43) KMT2AMEN1RAB9AUSP2ALDH1A1
SCHEMBL11239680 0.80 SLC6A2 (0.46) ALDH1A1MAPK1
Bromide SCHEMBL11471759 0.79 SLC6A2 (0.45) ALDH1A1MAPK1
SCHEMBL11248843 0.78 ALDH1A1 (0.42) KMT2AMEN1RAB9AUSP2ALDH1A1
SCHEMBL11479620 0.78 CCR8 (0.44) KMT2AMEN1ALDH1A1S1PR2TET3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4198417-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US claimed
EP-0016261-B1 SPIRO(DIBENZ(B,F)OXEPIN-PIPERIDINES) AND METHODS OF PREPARING SAME HOECHST AKTIENGESELLSCHAFT (DE) 1982-12-29 EP disclosed
EP-0016261-A1 Spiro(dibenz(b,f)oxepin-piperidines) and methods of preparing same HOECHST AKTIENGESELLSCHAFT (DE) 1980-10-01 EP disclosed
US-4198417-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed
US-4198418-A ANALGESICS, TRANQUILIZERS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed