SCHEMBL11241754

SCHEMBL11241754

Cc1cccc(-c2cc(C(=O)O)c(=O)[nH]c2C(C)C)n1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SORT1 Q99523 7/20 0.40
KDM4E B2RXH2 3/20 0.39
GAA P10253 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 1/20 0.39
CDK5 Q00535 2/20 0.37
CDK5R1 Q15078 2/20 0.37
TGFBR1 P36897 4/20 0.37
CCR1 P32246 1/20 0.37
CCR8 P51685 1/20 0.37
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11251060 0.89 TGFBR1 (0.43) CDK5CDK5R1TGFBR1CCR1CCR8
SCHEMBL11239015 0.81 PDE3B (0.41) TGFBR1CCR1CCR8
SCHEMBL11242528 0.81 CCR1 (0.40) CDK5CDK5R1TGFBR1CCR1CCR8
SCHEMBL11235398 0.78 GAA (0.45) KDM4EGAAHPGDHSD17B10TGFBR1
SCHEMBL11242990 0.76 TGFBR1 (0.35) CDK5CDK5R1TGFBR1CCR1CCR8
SCHEMBL11231230 0.74 CCR1 (0.44) TGFBR1CCR1CCR8
SCHEMBL11238710 0.74 CDK5 (0.49) KDM4EGAAHPGDHSD17B10CDK5
SCHEMBL16277390 0.70 SORT1 (0.55) SORT1KDM4EHPGDHSD17B10TGFBR1
SCHEMBL7847744 0.68 KDM4E (0.56) SORT1KDM4EHPGDHSD17B10TGFBR1
SCHEMBL6609571 0.67 ALDH1A1 (0.58) SORT1KDM4EHPGDTGFBR1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4312875-A 5-(Pyridinyl)-6-(lower-alkyl)-2(1H)-pyridinones, 1,2-dihydro-2-oxo-5-(pyridinyl)-6-(lower-alkyl)nicotinic acids and lower-alkyl esters thereof, and cardiotonic use thereof STERLING DRUG INC. (US) 1982-01-26 US disclosed