SCHEMBL11242290

SCHEMBL11242290

CCNc1cc(-c2ccc(C)cn2)c(C)[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.39
CCR5 P51681 1/20 0.39
CCR8 P51685 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PTGS2 P35354 3/20 0.36
METAP2 P50579 1/20 0.34
IRAK4 Q9NWZ3 2/20 0.34
CSF1R P07333 2/20 0.34
FLT3 P36888 2/20 0.34
PDGFRA P16234 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
USP2 O75604 1/20 0.33
CASP1 P29466 1/20 0.33
BRCA1 P38398 1/20 0.33
CASP7 P55210 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2A6 P11509 1/20 0.33
PDE9A O76083 1/20 0.33
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11231370 0.76 PDE3B (0.54) CCR1CCR5CCR8HDAC6PTGS2
SCHEMBL11248742 0.76 CCR1 (0.44) CCR1CCR5CCR8HDAC6PTGS2
SCHEMBL11239007 0.74 PDE3B (0.58) KMT2AMAPT
SCHEMBL11240175 0.73 PDE3A (0.57) CCR1CCR5CCR8HDAC6PTGS2
SCHEMBL11248993 0.73 GAA (0.50) CCR1CCR5CCR8HDAC6PTGS2
SCHEMBL11236627 0.72 CCR1 (0.40) CCR1CCR5CCR8HDAC6PTGS2
SCHEMBL11248533 0.69 CCR1 (0.50) CCR1CCR5CCR8HDAC6PTGS2
SCHEMBL11242267 0.69 TYRO3 (0.43) FLT3SMN1; SMN2
SCHEMBL2674107 0.65 P4HA1 (0.47) NPC1RAB9ASMN1; SMN2MAPTTP53
SCHEMBL11242990 0.63 TGFBR1 (0.35) CCR1CCR8METAP2IRAK4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed