SCHEMBL11242994

SCHEMBL11242994

CC(=O)N1CCC(C(=O)O)(c2ccccc2Oc2ccccc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.45
ALDH1A1 P00352 6/20 0.44
CYP2C19 P33261 3/20 0.44
MAPK1 P28482 2/20 0.44
MMP2 P08253 2/20 0.43
MMP9 P14780 2/20 0.43
TSHR P16473 4/20 0.43
CYP2D6 P10635 3/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
RAB9A P51151 1/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2C9 P11712 2/20 0.42
HSD17B10 Q99714 2/20 0.41
CYP1A2 P05177 1/20 0.41
HPGD P15428 1/20 0.41
ALOX12 P18054 1/20 0.41
HIF1A Q16665 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11241289 0.93 KMT2A (0.44) USP2ALDH1A1CYP2C19MAPK1MMP2
SCHEMBL11486442 0.92 USP2 (0.45) USP2ALDH1A1CYP2C19MAPK1MMP2
SCHEMBL11471965 0.90 MEN1 (0.43) USP2ALDH1A1CYP2C19MAPK1MMP2
SCHEMBL11244293 0.90 CYP2D6 (0.43) USP2ALDH1A1CYP2C19MAPK1MMP2
SCHEMBL5498370 0.84 CTNNB1 (0.46) ALDH1A1TSHRKMT2AMEN1HSD17B10
SCHEMBL11243000 0.82 USP2 (0.43) USP2ALDH1A1CYP2C19MAPK1MMP2
SCHEMBL11468367 0.80 SCN1A (0.48) ALDH1A1TSHRKMT2AMEN1CYP3A4
SCHEMBL11255002 0.80 OPRM1 (0.45) ALDH1A1KCNH2
SCHEMBL11479620 0.79 CCR8 (0.44) ALDH1A1KMT2AMEN1MAPTTET3
SCHEMBL11246081 0.79 MMP1 (0.45) ALDH1A1MMP9KMT2AMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4198417-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US claimed
EP-0016261-B1 SPIRO(DIBENZ(B,F)OXEPIN-PIPERIDINES) AND METHODS OF PREPARING SAME HOECHST AKTIENGESELLSCHAFT (DE) 1982-12-29 EP disclosed
EP-0016261-A1 Spiro(dibenz(b,f)oxepin-piperidines) and methods of preparing same HOECHST AKTIENGESELLSCHAFT (DE) 1980-10-01 EP disclosed
US-4198418-A ANALGESICS, TRANQUILIZERS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed
US-4198417-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed