SCHEMBL11246081

SCHEMBL11246081

CN1CCC(C(=O)O)(c2ccccc2Oc2ccc(Cl)cc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.45
MMP9 P14780 1/20 0.45
MMP13 P45452 1/20 0.45
ADAM17 P78536 1/20 0.45
OPRM1 P35372 4/20 0.44
SCN1A P35498 1/20 0.42
SCN2A Q99250 1/20 0.42
SCN3A Q9NY46 1/20 0.42
KCNH2 Q12809 2/20 0.41
SLC22A1 O15245 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
CCR8 P51685 1/20 0.41
RECQL P46063 1/20 0.40
LIPE Q05469 1/20 0.40
CHRM5 P08912 2/20 0.39
CHRM3 P20309 2/20 0.39
CHRM1 P11229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11255002 0.89 OPRM1 (0.45) OPRM1SCN1ASCN2ASCN3AKCNH2
SCHEMBL11479620 0.86 CCR8 (0.44) KCNH2CCR8KMT2AMAPTPNLIP
SCHEMBL11246085 0.83 MMP1 (0.43) MMP1MMP9MMP13ADAM17OPRM1
SCHEMBL11468367 0.82 SCN1A (0.48) OPRM1SCN1ASCN2ASCN3AKCNH2
Oxalic Acid SCHEMBL11468650 0.80 SCN1A (0.46) OPRM1SCN1ASCN2ASCN3AKCNH2
SCHEMBL11471019 0.80 SCN1A (0.46) OPRM1SCN1ASCN2ASCN3AKCNH2
SCHEMBL11478119 0.79 OPRM1 (0.48) OPRM1SCN1ASCN2ASCN3AKCNH2
SCHEMBL11242994 0.79 USP2 (0.45) MMP9KCNH2CCR8KMT2AMAPT
SCHEMBL5498370 0.78 CTNNB1 (0.46) KMT2AMAPTALDH1A1LMNAHPGD
Oxalic Acid SCHEMBL11471026 0.78 SCN1A (0.45) OPRM1SCN1ASCN2ASCN3AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4198417-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US claimed
EP-0016261-B1 SPIRO(DIBENZ(B,F)OXEPIN-PIPERIDINES) AND METHODS OF PREPARING SAME HOECHST AKTIENGESELLSCHAFT (DE) 1982-12-29 EP disclosed
EP-0016261-A1 Spiro(dibenz(b,f)oxepin-piperidines) and methods of preparing same HOECHST AKTIENGESELLSCHAFT (DE) 1980-10-01 EP disclosed
US-4198417-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed
US-4198418-A ANALGESICS, TRANQUILIZERS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed