SCHEMBL11243779

SCHEMBL11243779

NC(c1ccncc1)c1ccccc1C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
KMT2A Q03164 4/20 0.46
TDP1 Q9NUW8 3/20 0.46
GAA P10253 1/20 0.46
ALOX15 P16050 1/20 0.42
MEN1 O00255 3/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KDM4C Q9H3R0 3/20 0.41
MAPT P10636 2/20 0.40
HDAC8 Q9BY41 1/20 0.40
KDM4E B2RXH2 5/20 0.40
NAPRT Q6XQN6 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
KDM6B O15054 1/20 0.40
KDM4A O75164 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11675001 0.88 ALDH1A1 (0.53) ALDH1A1KMT2ATDP1GAAALOX15
SCHEMBL30251446 0.81 ALDH1A1 (0.47) ALDH1A1KMT2ATDP1GAAALOX15
SCHEMBL3168094 0.78 NAPRT (0.39) ALDH1A1KMT2ATDP1GAAALOX15
SCHEMBL3831520 0.75 BCAT2 (0.46) ALDH1A1KMT2ATDP1GAANPC1
SCHEMBL1449566 0.74 ALDH1A1 (0.52) ALDH1A1KMT2ATDP1GAAALOX15
SCHEMBL6372852 0.74 ALDH1A1 (0.56) ALDH1A1KMT2ATDP1GAAALOX15
SCHEMBL3998608 0.73 SLC6A3 (0.65) ALDH1A1KMT2AGAASLC6A2SLC6A4
SCHEMBL4758132 0.73 SLC6A3 (0.65) ALDH1A1KMT2AGAASLC6A2SLC6A4
SCHEMBL6436789 0.73 SLC6A3 (0.65) ALDH1A1KMT2AGAASLC6A2SLC6A4
SCHEMBL2906291 0.73 SLC6A3 (0.56) ALDH1A1KMT2ATDP1GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4309541-A CHEMICAL INTERMEDIATES TO QUINAZOLINE HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1982-01-05 US disclosed
US-4255429-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1981-03-10 US disclosed
EP-0009465-A1 N-(1-(4-amino-2-quinazolinyl)-3 or 4-piperidyl lactames, process for their preparation and pharmaceutical compositions containing them CIBA-GEIGY AG (CH) 1980-04-02 EP disclosed
US-4000287-A HYPOTENSIVES, ANTIARRHYTHMIC CIBA-GEIGY CORPORATION (US) 1976-12-28 US disclosed