SCHEMBL2906291

SCHEMBL2906291

O=C(O)c1ccccc1C(Cc1ccncc1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 2/20 0.56
SLC6A4 P31645 2/20 0.56
SLC6A2 P23975 1/20 0.56
LMNA P02545 3/20 0.47
CHRM1 P11229 2/20 0.45
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.43
KMT2A Q03164 2/20 0.43
TSHR P16473 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 1/20 0.43
NR3C2 P08235 2/20 0.43
CYP3A4 P08684 2/20 0.43
KDM4C Q9H3R0 2/20 0.41
EPHX2 P34913 1/20 0.41
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28205347 0.89 ALDH1A1 (0.49) SLC6A3SLC6A4SLC6A2ALDH1A1GAA
SCHEMBL29167634 0.78 SLC6A3 (0.88) SLC6A3SLC6A4SLC6A2LMNACHRM1
Iodide SCHEMBL3429365 0.76 SLC6A4 (0.84) SLC6A3SLC6A4SLC6A2LMNACHRM1
SCHEMBL5428376 0.75 ALDH1A1 (0.51) LMNAALDH1A1GAAKMT2ATSHR
SCHEMBL30251446 0.74 ALDH1A1 (0.47) SLC6A3SLC6A4SLC6A2ALDH1A1GAA
SCHEMBL27935564 0.74 HTR2A (0.54) ALDH1A1GAAKMT2ATDP1KDM4E
SCHEMBL8944151 0.74 ALDH1A1 (0.50) ALDH1A1GAAKMT2ATDP1KDM4E
SCHEMBL11243779 0.73 ALDH1A1 (0.46) SLC6A3SLC6A4SLC6A2ALDH1A1GAA
SCHEMBL29173215 0.73 SLC6A4 (1.00) SLC6A3SLC6A4SLC6A2LMNATSHR
SCHEMBL7816162 0.72 CHRM1 (0.61) SLC6A3SLC6A4SLC6A2LMNACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2216327-A1 Benzoic acid (1-phenyl-2-pyridin-4-yl)ethyl esters as phosphodiesterase inhibitors CHIESI FARMACEUTICI S.p.A. (IT) 2010-08-11 EP disclosed