SCHEMBL11244119

SCHEMBL11244119

Nc1cnc(NCCCS(N)(=O)=O)nc1O

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.32
CA2 P00918 6/20 0.32
CA9 Q16790 6/20 0.32
CA12 O43570 2/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
CA14 Q9ULX7 1/20 0.30
PDCD1 Q15116 1/20 0.30
CD274 Q9NZQ7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11154337 0.80 NUDT1 (0.44)
SCHEMBL11240946 0.79 SYK (0.35)
SCHEMBL10996367 0.79 TLR8 (0.43) MEN1ALDH1A1MAPTMAPK1RAB9A
SCHEMBL11399515 0.77 GAA (0.41) MEN1ALDH1A1GAAMAPK1KMT2A
SCHEMBL10998571 0.77 KMT2A (0.43) KMT2A
SCHEMBL11002056 0.77 KMT2A (0.43) KMT2A
SCHEMBL11236452 0.75 KCNH3 (0.43) MAPT
SCHEMBL11249857 0.75 MRGPRX1 (0.38) CA1CA2CA9CA12CA14
SCHEMBL10998512 0.75 MAPT (0.37) CA1CA2CA9MEN1ALDH1A1
SCHEMBL11391206 0.74 KDM4E (0.36) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0016374-B1 PENICILLINS, THEIR SALTS, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC AGENTS CONTAINING THESE COMPOUNDS Dr. Karl Thomae GmbH (DE) 1982-03-03 EP disclosed
US-4289775-A BACTERICIDAL ANTIBIOTICS KARL THOMAE GMBH (DE) 1981-09-15 US disclosed
EP-0016374-A1 Penicillins, their salts, process for their preparation and therapeutic agents containing these compounds Dr. Karl Thomae GmbH (DE) 1980-10-01 EP disclosed