SCHEMBL11246111

SCHEMBL11246111

COc1ccccc1-n1ccc(=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.59
TUBB4A P04350 1/20 0.49
TUBB P07437 1/20 0.49
TUBA3C P0DPH7 1/20 0.49
TUBA1B P68363 1/20 0.49
TUBA4A P68366 1/20 0.49
TUBB4B P68371 1/20 0.49
TUBB3 Q13509 1/20 0.49
TUBB2A Q13885 1/20 0.49
TUBB8 Q3ZCM7 1/20 0.49
TUBA3E Q6PEY2 1/20 0.49
TUBA1A Q71U36 1/20 0.49
TUBA1C Q9BQE3 1/20 0.49
TUBB6 Q9BUF5 1/20 0.49
TUBB2B Q9BVA1 1/20 0.49
TUBB1 Q9H4B7 1/20 0.49
GAA P10253 3/20 0.47
MAPT P10636 5/20 0.45
ALDH1A1 P00352 3/20 0.45
HPGD P15428 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2098026 0.84 CA12 (0.52) MGLLTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL29439366 0.74 MGLL (1.00) MGLLGAAMAPTALDH1A1MEN1
SCHEMBL141734 0.74 MGLL (1.00) MGLLGAAMAPTALDH1A1MEN1
SCHEMBL10916413 0.74 MGLL (0.55) MGLLTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL6559666 0.73 TUBB4A (0.49) MGLLTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL12841493 0.72 MEN1 (0.49) MGLLGAAMAPTALDH1A1HPGD
SCHEMBL7981999 0.72 GAA (0.58) MGLLGAAMAPTALDH1A1HPGD
SCHEMBL20917333 0.72 TUBB4A (0.65) MGLLTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL28842652 0.71 MGLL (0.57) MGLLGAAALDH1A1KMT2AKDM4E
SCHEMBL31149024 0.70 CYP19A1 (0.67) GAAMAPTALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0006628-B1 SUBSTITUTED DIHYDROPYRIDINE UREAS, PROCESS FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM MERCK & CO. INC. (US) 1982-12-29 EP disclosed
EP-0006628-A1 Substituted dihydropyridine ureas, process for preparing the same and pharmaceutical compositions containing them MERCK & CO. INC. (US) 1980-01-09 EP disclosed
US-4176187-A HYPOTENSIVE AGENTS MERCK & CO., INC. (US) 1979-11-27 US disclosed