SCHEMBL11247880

SCHEMBL11247880

CCc1nc(NC)c(C#N)cc1-c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
MAPK1 P28482 3/20 0.45
HSD17B10 Q99714 3/20 0.45
TSHR P16473 2/20 0.45
HPGD P15428 4/20 0.44
KDM4E B2RXH2 4/20 0.44
LMNA P02545 2/20 0.44
CLK1 P49759 1/20 0.44
CYP11B1 P15538 3/20 0.43
CYP11B2 P19099 3/20 0.43
ADORA1 P30542 2/20 0.43
MAPT P10636 2/20 0.42
HIF1A Q16665 1/20 0.42
PGK1 P00558 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ADORA2A P29274 1/20 0.40
KDM5A P29375 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
XDH P47989 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11226168 0.82 ALDH1A1 (0.49) ALDH1A1MAPK1HSD17B10TSHRHPGD
SCHEMBL11241191 0.78 WNT3A (0.45) CYP3A4
SCHEMBL11159205 0.77 MKNK1 (0.50) LMNAKMT2ACYP1A2CYP3A4CYP2C19
SCHEMBL11248371 0.74 CHEK1 (0.47) ALDH1A1HSD17B10HPGDKDM4ELMNA
SCHEMBL10841297 0.73 ALDH1A1 (0.45) ALDH1A1HSD17B10HPGDKDM4ELMNA
SCHEMBL11245356 0.70 CYP2A6 (0.44) ALDH1A1MAPK1HSD17B10TSHRCYP11B1
SCHEMBL2598836 0.70 CYP11B1 (0.53) ALDH1A1HPGDKDM4ECYP11B1CYP11B2
SCHEMBL10707484 0.69 PDE3B (0.73) ALDH1A1TSHRHPGDKDM4ELMNA
SCHEMBL7272652 0.69 CYP2A6 (0.47) ALDH1A1MAPK1HSD17B10TSHRCYP11B1
SCHEMBL11251403 0.68 PDE3B (0.50) ALDH1A1TSHRHPGDKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362734-A 2-(Substituted-amino)-5-(pyridinyl-nicotinonitriles, and their cardiotonic use STERLING DRUG INC. (US) 1982-12-07 US disclosed