SCHEMBL11248019

SCHEMBL11248019

O=C(O)Cc1c(C2CCCCC2)nn(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
P2RX7 Q99572 1/20 0.43
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
LMNA P02545 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
PKM P14618 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CFTR P13569 2/20 0.38
PTGDR2 Q9Y5Y4 2/20 0.38
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11245176 0.92 P2RX7 (0.44) CYP1A2CYP2C9CYP2C19P2RX7CNR1
SCHEMBL11251356 0.91 CYP1A2 (0.42) CYP1A2CYP2C9CYP2C19P2RX7CNR1
SCHEMBL11249532 0.86 ALDH1A1 (0.46) CYP1A2CYP2C9CYP2C19P2RX7CNR1
Trifezolac SCHEMBL11182574 0.76 KDM4E (0.51) CYP1A2CYP2C9CYP2C19LMNATP53
SCHEMBL6123601 0.75 CYP2C9 (0.51) CYP1A2CYP2C9CYP2C19CNR1CNR2
SCHEMBL1195159 0.75 CYP2C9 (0.62) CYP1A2CYP2C9CYP2C19P2RX7NPC1
SCHEMBL11247967 0.70 CYP2C9 (0.56) CYP1A2CYP2C9CYP2C19P2RX7LMNA
SCHEMBL11254239 0.70 CNR1 (0.47) CNR1CNR2PTGDR2
SCHEMBL11699362 0.70 KDM4E (0.55) CYP1A2CYP2C9CYP2C19L3MBTL1PTGDR2
SCHEMBL11254211 0.68 CA1 (0.53) CYP1A2CYP2C9CYP2C19CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4325962-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIDYRETICS BYK-GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1982-04-20 US disclosed
US-4146721-A ANALGESICS, ANTIINFLAMMATORY AGENTS AND ANTIPYRETICS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1979-03-27 US disclosed
US-4011332-A RODENTICIDE BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DT) 1977-03-08 US disclosed