SCHEMBL11248931

SCHEMBL11248931

N#CCc1cccc2c(-c3ccc(Cl)cc3)nccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 3/20 0.44
IDO1 P14902 1/20 0.44
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
CYP2A6 P11509 1/20 0.35
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
ERBB2 P04626 1/20 0.34
HPGD P15428 1/20 0.34
GRIA1 P42261 1/20 0.34
CACNG8 Q8WXS5 1/20 0.34
NR4A2 P43354 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11263093 0.87 TDO2 (0.41) TDO2PDE3BPDE3AKMT2AMEN1
SCHEMBL11253084 0.86 ALDH1A1 (0.36) TDO2KMT2AMEN1CYP1A2CYP2C19
SCHEMBL11261674 0.86 TDO2 (0.36) TDO2IDO1KMT2AMEN1CYP1A2
SCHEMBL11251011 0.86 BCHE (0.44) TDO2PDE3BPDE3AALDH1A1ERBB2
SCHEMBL11261938 0.83 ALDH1A1 (0.43) PDE3BPDE3AKMT2AMEN1ALDH1A1
SCHEMBL11252484 0.83 HSP90AA1 (0.35) TDO2ALDH1A1
SCHEMBL11254978 0.83 SYK (0.35) TDO2KMT2AMEN1CYP1A2CYP2C9
SCHEMBL11254049 0.83 TDO2 (0.37) TDO2NPSR1KDM4E
SCHEMBL11262405 0.82 TDO2 (0.48) TDO2IDO1PDE3BPDE3AKMT2A
SCHEMBL11256404 0.81 TDO2 (0.47) TDO2IDO1PDE3BPDE3AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed