SCHEMBL11261674

SCHEMBL11261674

N#CCc1cccc2c(-c3ccc(Br)cc3)nccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 3/20 0.36
CSNK2A1 P68400 2/20 0.35
ERBB2 P04626 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
IDO1 P14902 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
TNF P01375 1/20 0.32
PTGES O14684 1/20 0.32
GPR84 Q9NQS5 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11263093 0.87 TDO2 (0.41) TDO2ADORA2AALDH1A1NPSR1MEN1
SCHEMBL11253084 0.86 ALDH1A1 (0.36) TDO2ERBB2ADORA2AADORA1ALDH1A1
SCHEMBL11251011 0.86 BCHE (0.44) TDO2ERBB2ADORA2AADORA1ALDH1A1
SCHEMBL11248931 0.86 TDO2 (0.44) TDO2ERBB2IDO1ALDH1A1CYP1A2
SCHEMBL11254978 0.83 SYK (0.35) TDO2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL11254049 0.83 TDO2 (0.37) TDO2NPSR1
SCHEMBL11252484 0.83 HSP90AA1 (0.35) TDO2ALDH1A1TNFCYP11B1CYP11B2
SCHEMBL11261938 0.83 ALDH1A1 (0.43) ADORA2AADORA1ALDH1A1NPSR1MEN1
SCHEMBL11249519 0.82 NPC1 (0.43) TDO2IDO1ALDH1A1CYP1A2CYP3A4
SCHEMBL11258335 0.82 ALDH1A1 (0.39) TDO2IDO1ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed