SCHEMBL11256404

SCHEMBL11256404

Clc1ccc(-c2nccc3c(CBr)cccc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 2/20 0.47
IDO1 P14902 2/20 0.47
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
KMT2A Q03164 4/20 0.38
NPSR1 Q6W5P4 3/20 0.38
GAA P10253 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
MEN1 O00255 2/20 0.38
CSNK2A2 P19784 1/20 0.37
CSNK2B P67870 1/20 0.37
ALDH1A1 P00352 3/20 0.36
LMNA P02545 3/20 0.36
HPGD P15428 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
HTT P42858 1/20 0.36
CRHR1 P34998 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11262405 0.86 TDO2 (0.48) TDO2IDO1PDE3BPDE3AKMT2A
SCHEMBL11256693 0.86 ALDH1A1 (0.39) TDO2IDO1KMT2ANPSR1GAA
SCHEMBL11253962 0.82 TDO2 (0.45) TDO2IDO1PDE3BPDE3AKMT2A
SCHEMBL11248931 0.81 TDO2 (0.44) TDO2IDO1PDE3BPDE3AKMT2A
SCHEMBL11255704 0.80 PTGDR2 (0.49) TDO2IDO1PDE3BPDE3AKMT2A
SCHEMBL11248945 0.79 IDO1 (0.42) TDO2IDO1PDE3BPDE3AKMT2A
SCHEMBL11500393 0.78 PTGDR2 (0.45) TDO2IDO1KMT2ACYP1A2CYP2C9
SCHEMBL11258335 0.77 ALDH1A1 (0.39) TDO2IDO1KMT2ANPSR1GAA
SCHEMBL11260499 0.76 TDO2 (0.50) TDO2IDO1PDE3BPDE3AKMT2A
SCHEMBL11266566 0.76 KDR (0.40) TDO2IDO1PDE3BPDE3AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed